SCHEMBL4752018

SCHEMBL4752018

O=C1OC(=O)C(c2ccc(OC=S)cc2)=C1c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.49
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MITF O75030 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HPGD P15428 1/20 0.36
NTSR1 P30989 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PTGS1 P23219 2/20 0.36
PDE4B Q07343 1/20 0.35
GSTP1 P09211 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
NR1H2 P55055 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4788888 0.81 PTGS2 (0.50) PTGS2HPGD
SCHEMBL10736364 0.79 PTGS2 (0.69) PTGS2KMT2AMEN1MAPTKDM4E
SCHEMBL4787548 0.78 PTGS2 (0.60) PTGS2KMT2AMEN1MAPTALDH1A1
SCHEMBL592300 0.77 PTGS2 (0.65) PTGS2KMT2AMEN1MAPTKDM4E
SCHEMBL934950 0.72
Hydrochloric Acid SCHEMBL29124791 0.70 LTA4H (0.43) KMT2AMEN1ALDH1A1LMNACA1
SCHEMBL30320677 0.70 ME2 (0.57) PTGS2KMT2AMEN1MAPTALDH1A1
SCHEMBL6674116 0.67 PTGS2 (0.55) PTGS2KMT2AMEN1MAPTKDM4E
SCHEMBL10733826 0.67 PTGS2 (0.55) PTGS2MAPT
SCHEMBL27521616 0.67 PTGS2 (0.46) PTGS2KMT2AMEN1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO claimed
WO-2008140251-A2 CYCLOOXYGENASE-2 INHIBITORS UNIVERSITY-INDUSTRY COOPERATION GROUP OF KYUNG HEE UNIVERSITY (KR) 2008-11-20 WO disclosed