SCHEMBL4788710

SCHEMBL4788710

Cc1c(C(=O)N[C@@H]2CCc3cccc(N4CCN(C)CC4)c3C2)nnn1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.50
NPY5R Q15761 1/20 0.43
ROCK1 Q13464 1/20 0.42
KCNH2 Q12809 4/20 0.42
SCN5A Q14524 4/20 0.42
SCN9A Q15858 4/20 0.42
CCR1 P32246 1/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GPR52 Q9Y2T5 1/20 0.39
MAPT P10636 3/20 0.39
THRB P10828 1/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789431 0.86 SCN9A (0.60) SMN1; SMN2ROCK1KCNH2SCN5ASCN9A
SCHEMBL7031232 0.81 MEN1 (0.55) KCNH2SCN5ASCN9AMEN1KMT2A
SCHEMBL7030282 0.81 MEN1 (0.55) KCNH2SCN5ASCN9AMEN1KMT2A
SCHEMBL2079393 0.81 SMN1; SMN2 (0.62) SMN1; SMN2NPY5RROCK1CCR1KDM4E
SCHEMBL4788895 0.81 KCNH2 (0.49) KCNH2SCN5ASCN9AMEN1KMT2A
SCHEMBL6820338 0.79 KCNH2 (0.55) SMN1; SMN2KCNH2SCN5ASCN9AMEN1
SCHEMBL6820334 0.79 KCNH2 (0.55) SMN1; SMN2KCNH2SCN5ASCN9AMEN1
SCHEMBL7025761 0.79 KCNH2 (0.55) SMN1; SMN2KCNH2SCN5ASCN9AMEN1
SCHEMBL4789479 0.78 LCK (0.46) KCNH2SCN5ASCN9AKDM4EMEN1
SCHEMBL2079395 0.78 LMNA (0.58) SMN1; SMN2NPY5RROCK1CCR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO claimed
WO-2008130321-A2 NOVEL N-TETRAHYDRONAPHTALENE OR 5-HETEROCYCLYL-CHROMANE OR 8-HETEROCYCLYL-TETRAHYDRONAPHTALENE DERIVATIVES FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2008-10-30 WO disclosed