SCHEMBL4789663

SCHEMBL4789663

NC(=O)c1c[nH]c2c1CCC2=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.38
CSNK1A1 P48729 1/20 0.38
LIMK1 P53667 1/20 0.38
MAP2K1 Q02750 1/20 0.38
PRKAA1 Q13131 1/20 0.38
DYRK1A Q13627 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
BRD4 O60885 1/20 0.38
ALDH1A1 P00352 1/20 0.37
ATM Q13315 1/20 0.37
NNMT P40261 2/20 0.34
AURKA O14965 1/20 0.33
PARP1 P09874 1/20 0.33
PIM1 P11309 1/20 0.30
PIM3 Q86V86 1/20 0.30
ALOX15 P16050 1/20 0.30
MAPK1 P28482 1/20 0.30
CASP1 P29466 1/20 0.30
CASP7 P55210 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12466646 0.77 MAP2K1 (0.45) MAP2K1ATM
SCHEMBL3604129 0.71 SIRT3 (0.43) NNMT
SCHEMBL12466445 0.70 NNMT (0.38) NNMTAURKAPIM1
SCHEMBL31297123 0.68 NTRK1 (0.46) CSNK1A1DYRK1BBRD4ALDH1A1ATM
SCHEMBL4789593 0.68 HSD17B10 (0.47) BRD4ALDH1A1ATMNNMTPARP1
SCHEMBL26110395 0.68 HSD17B10 (0.44) CSNK1A1DYRK1BBRD4ALDH1A1ATM
SCHEMBL12466356 0.68 PIM1 (0.39) NNMTAURKAPIM1
SCHEMBL7394232 0.64 ALDH1A1 (0.39) MAPK8CSNK1A1LIMK1MAP2K1PRKAA1
SCHEMBL21471348 0.64 PARP1 (0.53) BRD4ALDH1A1AURKAPARP1ALOX15
SCHEMBL8362799 0.64 MAPT (0.42) ALDH1A1ATMNNMTPARP1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008148034-A1 MAPK/ERK KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-12-04 WO claimed
WO-2008148034-A1 MAPK/ERK KINASE INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-12-04 WO disclosed