SCHEMBL4789958

SCHEMBL4789958

NC(=O)c1cccc(-c2cccnc2)c1Oc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.47
BCAT2 O15382 1/20 0.46
PKN1 Q16512 1/20 0.46
PKN2 Q16513 1/20 0.46
MKNK1 Q9BUB5 9/20 0.46
MKNK2 Q9HBH9 8/20 0.46
MAPK8 P45983 1/20 0.45
MAPK10 P53779 1/20 0.45
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44
JAK2 O60674 1/20 0.44
JAK3 P52333 1/20 0.44
PARP1 P09874 1/20 0.44
DHODH Q02127 1/20 0.44
PARP2 Q9UGN5 1/20 0.44
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28081509 0.87 BCAT2 (0.61) CTNNB1BCAT2ALDH1A1PARP1KDM4E
SCHEMBL4789960 0.81 CTNNB1 (0.56) CTNNB1PKN1PKN2MKNK1MKNK2
SCHEMBL167082 0.80 BCAT2 (0.67) BCAT2PKN1PKN2MKNK1MKNK2
SCHEMBL31227976 0.80 BCAT2 (0.67) BCAT2PKN1PKN2MKNK1MKNK2
SCHEMBL30514275 0.80 BCAT2 (0.67) BCAT2PKN1PKN2MKNK1MKNK2
SCHEMBL28131715 0.79 ALDH1A1 (0.47) CTNNB1MKNK1MKNK2ALDH1A1MAPK1
Hydrochloric Acid SCHEMBL27890957 0.78 BCAT2 (0.65) BCAT2PKN1PKN2MKNK1MKNK2
Hydrochloric Acid SCHEMBL30165666 0.78 BCAT2 (0.65) BCAT2PKN1PKN2MKNK1MKNK2
SCHEMBL3717538 0.78 CA12 (0.43) ALDH1A1HSD17B10KDM4ELMNA
SCHEMBL8809860 0.78 BCAT2 (0.56) BCAT2PKN1PKN2MKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957073-A2 MEDICINAL DRUG OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-08-20 EP disclosed
WO-2007066784-A2 DIARYLETHER DERIVATIVES AS ANTITUMOR AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-06-14 WO disclosed