SCHEMBL4790306

SCHEMBL4790306

CS(=O)(=O)c1ccc2c(c1)CCN(C(=O)C1CCCCC1C(=O)NC1(C#N)CC1)C2

nearest known ligand 0.69

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 19/20 0.69
CTSB P07858 9/20 0.66
CTSS P25774 5/20 0.66
CTSL P07711 1/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C9 P11712 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105820 0.89 CTSK (0.57) CTSKCTSBCTSS
SCHEMBL4789905 0.89 CTSK (0.57) CTSKCTSBCTSS
SCHEMBL4789866 0.84 CTSK (0.70) CTSKCTSBCTSSCTSL
SCHEMBL8100014 0.82 CTSK (0.60) CTSKCTSBCTSS
SCHEMBL2241411 0.82 CTSK (1.00) CTSKCTSBCTSS
SCHEMBL2243628 0.82 CTSK (1.00) CTSKCTSBCTSS
SCHEMBL4788694 0.81 CTSK (0.67) CTSKCTSBCTSS
SCHEMBL8121853 0.81 CTSK (0.67) CTSKCTSBCTSS
SCHEMBL8107252 0.81 CTSK (0.67) CTSKCTSBCTSS
SCHEMBL8111299 0.81 CTSK (0.67) CTSKCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001128-A1 1,2-CYCL0HEXANE DICARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed