SCHEMBL8100014

SCHEMBL8100014

N#CC1(NC(=O)[C@@H]2CCCC[C@H]2C(=O)N2CCc3cc(F)c(F)cc3C2)CC1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSK P43235 19/20 0.60
CTSB P07858 3/20 0.60
CTSS P25774 2/20 0.59
KCNH2 Q12809 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8107252 0.89 CTSK (0.67) CTSKCTSBCTSSKCNH2
SCHEMBL8111299 0.87 CTSK (0.67) CTSKCTSBCTSSKCNH2
SCHEMBL4788694 0.87 CTSK (0.67) CTSKCTSBCTSSKCNH2
SCHEMBL4789866 0.85 CTSK (0.70) CTSKCTSBCTSSKCNH2
SCHEMBL8121853 0.85 CTSK (0.67) CTSKCTSBCTSSKCNH2
SCHEMBL4787930 0.84 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL8109032 0.84 CTSK (0.69) CTSKCTSBCTSSKCNH2
SCHEMBL4790306 0.82 CTSK (0.69) CTSKCTSBCTSS
SCHEMBL8105739 0.82 CTSK (0.62) CTSKCTSBCTSSKCNH2
SCHEMBL8100091 0.82 CTSK (0.62) CTSKCTSBCTSSKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009001128-A1 1,2-CYCL0HEXANE DICARBOXAMIDES AS CATHEPSIN INHIBITORS ASTRAZENECA AB (SE) 2008-12-31 WO disclosed