SCHEMBL4790429

SCHEMBL4790429

COCC(=O)Nc1ccccc1-c1c[nH]cn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.52
GAA P10253 1/20 0.48
MAPT P10636 4/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
LMNA P02545 2/20 0.47
KDM4E B2RXH2 3/20 0.46
HSD17B10 Q99714 2/20 0.46
BDKRB1 P46663 1/20 0.46
ALDH1A1 P00352 5/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1906832 0.81 ALDH1A1 (0.50) GAAKDM4EHSD17B10ALDH1A1NPC1
SCHEMBL1950652 0.77 BRD9 (0.42) MAPTKMT2AMEN1LMNAMAPK10
SCHEMBL28006160 0.73 MAPT (0.40) MAPTKMT2AMEN1LMNAKDM4E
SCHEMBL9041899 0.70 KDM4E (0.62) TSHRGAAMAPTKMT2AMEN1
SCHEMBL1949655 0.70 KDM1A (0.48) L3MBTL1HTTMETAP2
SCHEMBL7547745 0.70 SMN1; SMN2 (0.71) TSHRGAAMAPTKMT2AMEN1
SCHEMBL27144018 0.70 TSHR (0.70) TSHRGAAMAPTKMT2AMEN1
SCHEMBL28006058 0.69 ALDH1A1 (0.36) TSHRMAPTKMT2AMEN1LMNA
SCHEMBL1905105 0.69 LMNA (0.41) LMNAKDM4EHSD17B10ALDH1A1L3MBTL1
SCHEMBL14818749 0.68 TSHR (0.68) TSHRGAAMAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966185-A2 2-AMINO-5-PIPERIDINYLIMIDAZOLONE COMPOUNDS AND USE THEREOF FOR ß-SECRETASE MODULATION Wyeth a Corporation of the State of Delaware (US) 2008-09-10 EP disclosed
WO-2007078813-A2 2-AMINO-5-PIPERIDINYLIMIDAZOLONE COMPOUNDS AND USE THEREOF FOR β-SECRETASE MODULATION WYETH (US) 2007-07-12 WO disclosed