SCHEMBL4790993

SCHEMBL4790993

COc1cccc(Oc2ccc([N+](=O)[O-])cc2Cl)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.71
HPGD P15428 4/20 0.71
ALDH1A1 P00352 7/20 0.65
MEN1 O00255 6/20 0.65
KMT2A Q03164 6/20 0.65
LMNA P02545 4/20 0.65
SMN1; SMN2 Q16637 4/20 0.65
PDE7A Q13946 1/20 0.60
GPR55 Q9Y2T6 1/20 0.57
GAA P10253 2/20 0.55
PKM P14618 1/20 0.55
NPSR1 Q6W5P4 2/20 0.54
HSP90AA1 P07900 1/20 0.54
NPC1 O15118 1/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
RAB9A P51151 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19399643 0.90 MAPT (0.61) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL3506576 0.87 PDE7A (0.66) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL2529627 0.86 ALDH1A1 (0.67) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL5315872 0.84 MAPT (0.67) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL4029870 0.84 PDE7A (0.73) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL3507438 0.83 MEN1 (0.65) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL8810667 0.83 PDE7A (0.72) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL4030285 0.83 MEN1 (0.61) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL3505754 0.83 MEN1 (0.61) MAPTHPGDALDH1A1MEN1KMT2A
SCHEMBL3506769 0.82 MAPT (0.60) MAPTHPGDALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110483366-B Indole compound and preparation method, pharmaceutical composition and application thereof 中国医学科学院药物研究所 2022-09-16 CN disclosed
EP-1957495-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-08-20 EP disclosed
WO-2007064045-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-07 WO disclosed