SCHEMBL4792188

SCHEMBL4792188

CN(C(=O)OCc1cc(Br)n(S(=O)(=O)c2cccnc2)c1)C(C)(C)C.CNC(=O)OCc1cc(-c2ccc(OC(F)F)cc2)n(S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGER4 P35408 1/20 0.32
NAMPT P43490 1/20 0.32
ADAM17 P78536 1/20 0.31
CYP3A4 P08684 2/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
MMP1 P03956 1/20 0.30
MMP9 P14780 1/20 0.30
MMP13 P45452 1/20 0.30
ELOVL6 Q9H5J4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4566466 0.82 RXFP1 (0.37) NAMPTADAM17MMP1MMP9MMP13
SCHEMBL2472672 0.79 NAMPT (0.43) NAMPTCYP3A4MMP1MMP9MMP13
SCHEMBL1278509 0.77 HTT (0.35) PTGER4ELOVL6
SCHEMBL1580484 0.76 CYP3A4 (0.39) PTGER4NAMPTCYP3A4CYP2C9CYP2C19
SCHEMBL3910397 0.76 DAGLA (0.40) PTGER4NAMPTMMP9
SCHEMBL1278511 0.74 DAGLA (0.38) PTGER4ELOVL6
SCHEMBL1278507 0.74 PTGER4 (0.38) PTGER4CYP3A4CYP2C9CYP2C19ELOVL6
Fumaric Acid SCHEMBL1278437 0.74 PTGER4 (0.39) PTGER4NAMPTCYP3A4CYP2C9CYP2C19
Fumaric Acid SCHEMBL1278433 0.74 PTGER4 (0.39) PTGER4NAMPTCYP3A4CYP2C9CYP2C19
SCHEMBL3910404 0.73 ALDH1A1 (0.41) PTGER4NAMPTCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed