SCHEMBL2472672

SCHEMBL2472672

CNC(=O)OCc1cc(Br)n(S(=O)(=O)c2cccnc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.43
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
HDAC1 Q13547 2/20 0.38
TSHR P16473 1/20 0.37
IDE P14735 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.36
TOP2A P11388 1/20 0.36
TOP2B Q02880 1/20 0.36
MMP1 P03956 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4566466 0.82 RXFP1 (0.37) NAMPTMAPTHDAC1TSHRIDE
SCHEMBL2415052 0.81 MEP1B (0.43) CYP3A4ALDH1A1KMT2AHDAC1
SCHEMBL19971357 0.80 IDE (0.39) NAMPTCYP3A4HTTHDAC1TSHR
SCHEMBL4792188 0.79 PTGER4 (0.32) NAMPTCYP3A4MMP1MMP9MMP13
SCHEMBL19971346 0.79 IDE (0.41) NAMPTMEN1KMT2AHDAC1IDE
SCHEMBL19971349 0.79 IDE (0.40) NAMPTHTTTSHRIDECHRNB4
SCHEMBL1157226 0.77 ALDH1A1 (0.49) NAMPTALDH1A1MEN1KMT2AHDAC1
SCHEMBL1157224 0.77 NAMPT (0.43) NAMPTALDH1A1LMNAKMT2AHDAC1
SCHEMBL2411499 0.77 ADAM17 (0.35) MEN1LMNAHTTKMT2AHDAC1
SCHEMBL1156490 0.77 ALDH1A1 (0.49) ALDH1A1MEN1LMNAKMT2AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed