SCHEMBL4792841

SCHEMBL4792841

CN(C)CCCNc1ncc2c(=O)c(C(=O)O)cn(-c3ccccc3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 10/20 0.47
KDM4E B2RXH2 1/20 0.42
MERTK Q12866 1/20 0.41
PDE4A P27815 1/20 0.40
KCNH2 Q12809 1/20 0.40
KMT2A Q03164 2/20 0.39
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
SLC2A1 P11166 1/20 0.38
APOBEC3A P31941 1/20 0.38
RAD52 P43351 1/20 0.38
RAB9A P51151 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3289880 0.93 CSF1R (0.56) CSF1RMERTK
SCHEMBL3293467 0.92 CSF1R (0.49) CSF1RKDM4EMERTKPDE4AKCNH2
SCHEMBL3289961 0.89 POLB (0.49) CSF1RKDM4EMERTKKMT2ANPC1
SCHEMBL11017743 0.88 CSF1R (0.49) CSF1RKDM4EPDE4AKCNH2
SCHEMBL4775328 0.85 CSF1R (0.68) CSF1R
SCHEMBL28527127 0.83 CSF1R (0.59) CSF1RKDM4EPDE4AKCNH2RAB9A
SCHEMBL4796017 0.81 CSF1R (0.59) CSF1RKDM4EMERTKKMT2ANPC1
SCHEMBL3293227 0.79 CSF1R (0.56) CSF1RMERTKPDE4AKCNH2KMT2A
SCHEMBL3291712 0.79 CSF1R (0.54) CSF1RKDM4EMERTKPDE4AKCNH2
SCHEMBL4773699 0.79 CSF1R (0.47) CSF1RKDM4EMERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945637-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-23 EP claimed
WO-2007033137-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO claimed