SCHEMBL4793153

SCHEMBL4793153

Cc1ccncc1-c1cc(CCC(C)(C)C)cn1S(=O)(=O)c1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.35
PTGES2 Q9H7Z7 1/20 0.35
CHRM5 P08912 1/20 0.34
PTGS2 P35354 4/20 0.34
HTR6 P50406 2/20 0.34
TSHR P16473 3/20 0.33
OPRM1 P35372 1/20 0.33
OPRK1 P41145 1/20 0.33
CNR2 P34972 2/20 0.33
NAPRT Q6XQN6 1/20 0.32
GAA P10253 1/20 0.32
GFER P55789 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790343 0.88 CYP2E1 (0.39) POLBCHRM5HTR6TSHRCNR2
SCHEMBL4792179 0.86 CYP2A6 (0.36) POLBCHRM5PTGS2TSHRCNR2
SCHEMBL1580390 0.83 TSHR (0.39) POLBPTGES2CHRM5PTGS2HTR6
SCHEMBL4793066 0.82 PTGS2 (0.40) PTGS2
SCHEMBL4791377 0.82 GBA1 (0.38) HTR6CNR2NAPRTSMN1; SMN2
SCHEMBL3906007 0.80 TSHR (0.42) TSHR
SCHEMBL1278515 0.79 NAMPT (0.40) HTR6TSHRGAAGFERSMN1; SMN2
SCHEMBL1278681 0.78 TACR1 (0.38) TSHRGAAGFERSMN1; SMN2
SCHEMBL4793151 0.78 PTGES2 (0.35) POLBPTGES2CHRM5PTGS2HTR6
Fumaric Acid SCHEMBL1278086 0.77 HDAC1 (0.36) POLBTSHRGAAGFERSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed