SCHEMBL4793151

SCHEMBL4793151

C[C](c1cc(-c2cnccc2C)n(S(=O)(=O)c2cccnc2)c1)C(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.35
NAPRT Q6XQN6 1/20 0.35
CHRM5 P08912 1/20 0.35
PTGS2 P35354 3/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR6 P50406 1/20 0.33
USP2 O75604 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
HDAC1 Q13547 1/20 0.32
CHRM1 P11229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4790340 0.88 CYP2A6 (0.42) NAPRTCHRM5KDM4EPOLBKMT2A
SCHEMBL4792177 0.85 CYP2A6 (0.37) NAPRTCHRM5PTGS2KDM4EPOLB
SCHEMBL4793065 0.82 PTGS2 (0.44) PTGS2
SCHEMBL4791372 0.81 GBA1 (0.40) NAPRTKDM4EPOLBKMT2AMAPT
SCHEMBL4793153 0.78 POLB (0.35) PTGES2NAPRTCHRM5PTGS2POLB
SCHEMBL1580390 0.75 TSHR (0.39) PTGES2CHRM5PTGS2POLBKMT2A
SCHEMBL3906007 0.75 TSHR (0.42) LMNA
SCHEMBL1278515 0.73 NAMPT (0.40) KDM4EHTR6LMNASMN1; SMN2
SCHEMBL1278681 0.73 TACR1 (0.38) KDM4EUSP2HTTNPSR1LMNA
Methylamine SCHEMBL28367776 0.73 PSEN1 (0.39) PTGES2NAPRTCHRM5PTGS2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919865-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2008-05-14 EP disclosed
WO-2007026916-A1 1-HETEROCYCLYLSULFONYL, 2-AMINOMETHYL, 5- (HETERO-) ARYL SUBSTITUTED 1-H-PYRROLE DERIVATIVES AS ACID SECRETION INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-03-08 WO disclosed