SCHEMBL4794530

SCHEMBL4794530

CCOCCN(C(=O)C1CCC(C)CC1)c1cc(-c2ccc(-c3cc4ncccn4n3)cc2)sc1C(=O)OC

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.35
HTT P42858 1/20 0.35
ATM Q13315 1/20 0.35
SYK P43405 2/20 0.34
MAPT P10636 4/20 0.33
TP53 P04637 1/20 0.33
ALDH1A1 P00352 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
PDE4D Q08499 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4794527 1.00 KDM4E (0.35) KDM4EHTTATMSYKMAPT
SCHEMBL4795067 0.94 ALDH1A1 (0.38) KDM4EHTTATMSYKMAPT
SCHEMBL4794496 0.94 CYP2E1 (0.34) SYKALDH1A1
SCHEMBL4794493 0.94 CYP2E1 (0.34) SYKALDH1A1
SCHEMBL4795076 0.94 ALDH1A1 (0.38) KDM4EHTTATMSYKMAPT
SCHEMBL4155397 0.91 KDM4E (0.38) KDM4EHTTATMSYKMAPT
SCHEMBL4155399 0.91 KDM4E (0.38) KDM4EHTTATMSYKMAPT
SCHEMBL4152953 0.88 KDM4E (0.37) KDM4EHTTATMSYKMAPT
SCHEMBL4152956 0.88 KDM4E (0.37) KDM4EHTTATMSYKMAPT
SCHEMBL4726531 0.88 ALDH1A1 (0.39) KDM4ESYKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008017688-A1 2-CARBOXY THIOPHENE DERIVATIVES AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-14 WO disclosed