SCHEMBL4795308

SCHEMBL4795308

[AsH2]c1nc(-c2ccccc2)c2nc(-c3ccc(N4CCNCC4)cc3)ccc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 4/20 0.51
PIM3 Q86V86 4/20 0.51
PIM2 Q9P1W9 3/20 0.51
MAP4K1 Q92918 2/20 0.47
KHK P50053 1/20 0.43
CETP P11597 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
ADRB1 P08588 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
KDM4E B2RXH2 3/20 0.41
HIF1A Q16665 2/20 0.41
S1PR2 O95136 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4112896 0.86 PIM1 (0.51) PIM1PIM3PIM2MAP4K1KHK
SCHEMBL4795298 0.83 HTR7 (0.51) ALDH1A1HPGDADRB1HTR3AKDM4E
SCHEMBL4106851 0.74 MAPT (0.55) PIM1MAP4K1ALDH1A1HPGDKDM4E
SCHEMBL12324749 0.72 KDM4E (0.72) PIM1PIM3PIM2CETPALDH1A1
SCHEMBL4110029 0.72 ATR (0.53) ALDH1A1HPGDHIF1AACVR1CYP1A2
SCHEMBL4112835 0.72 PIM1 (0.45) PIM1PIM3PIM2MAP4K1KHK
SCHEMBL4101654 0.71 ATR (0.53) KDM4EHIF1AS1PR2LMNAKMT2A
SCHEMBL1359864 0.71 ADRB1 (0.76) PIM1PIM3PIM2KHKCETP
SCHEMBL4112507 0.70 MAP4K1 (0.47) MAP4K1ALDH1A1KDM4ENPC1MAPT
SCHEMBL4112890 0.70 HTR7 (0.51) ALDH1A1HPGDADRB1KDM4EHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO disclosed