SCHEMBL480054

SCHEMBL480054

COc1ccc(C(C=O)c2cnc(C)cn2)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 1/20 0.37
ALDH1A1 P00352 2/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
JAK2 O60674 1/20 0.33
TYK2 P29597 1/20 0.33
HTR2A P28223 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
CRHR1 P34998 2/20 0.33
CYP1A2 P05177 1/20 0.33
POLB P06746 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
NFE2L2 Q16236 4/20 0.32
NPBWR1 P48145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL480170 0.78 DYRK1A (0.40) S1PR4NPSR1JAK2TYK2HTR2A
SCHEMBL27974261 0.77 ALDH1A1 (0.39) S1PR4ALDH1A1TSHRNPSR1HTR2A
SCHEMBL480065 0.73 NFE2L2 (0.39) NPSR1JAK2TYK2HTR2ASLC6A4
SCHEMBL479987 0.72 ALDH1A1 (0.46) ALDH1A1TSHRNPSR1CYP1A2POLB
SCHEMBL28034745 0.70 HTR2A (0.44) ALDH1A1JAK2TYK2HTR2ASLC6A4
SCHEMBL27974260 0.70 ALDH1A1 (0.44) S1PR4ALDH1A1TSHRNPSR1JAK2
SCHEMBL20550917 0.69 HTR2A (0.40) ALDH1A1JAK2TYK2HTR2ASLC6A4
SCHEMBL479926 0.68 KMT2A (0.36) ALDH1A1TSHRNPSR1HTR2ASLC6A4
SCHEMBL5188701 0.68 MAPT (0.44) ALDH1A1TSHRKCNH2HPGDL3MBTL1
SCHEMBL479938 0.68 ALDH1A1 (0.44) ALDH1A1TSHRNPSR1CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed
WO-2010108902-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2010-09-30 WO disclosed
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed