SCHEMBL480059

SCHEMBL480059

CC(c1ccc(-c2cccc(F)c2)cc1Cl)C(O)(c1cccc2cnccc12)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.38
TRPV1 Q8NER1 6/20 0.36
CYP11B2 P19099 4/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TNF P01375 2/20 0.33
PIP4K2A P48426 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
LMNA P02545 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
CYP11B1 P15538 3/20 0.32
CYP19A1 P11511 2/20 0.32
CYP17A1 P05093 1/20 0.32
CYP3A4 P08684 1/20 0.32
JAK2 O60674 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL837634 0.86 TRPV1 (0.38) TRPV1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL479777 0.86 TRPV1 (0.39) TRPV1CSNK2A2CSNK2BCYP3A4
SCHEMBL752272 0.86 TRPV1 (0.39) TRPV1CSNK2A2CSNK2BCYP3A4
SCHEMBL480188 0.85 KDM4E (0.36) TRPV1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL15789783 0.84 TRPV1 (0.38) TRPV1GPBAR1CYP3A4
SCHEMBL480178 0.84 TRPV1 (0.39) TRPV1
SCHEMBL734642 0.83 ALDH1A1 (0.37) TRPV1CYP11B2KDM4EALDH1A1MAPT
SCHEMBL480028 0.79 P2RX7 (0.36) TRPV1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL480023 0.74 MRGPRX4 (0.42) TRPV1SMN1; SMN2CYP3A4
SCHEMBL753267 0.74 MRGPRX4 (0.42) TRPV1SMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411361-A1 1,1,1-TRIFLUORO-2-HYDROXYPROPYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2012-02-01 EP disclosed