SCHEMBL4801731

SCHEMBL4801731

Cc1ccccc1C1NCCCn2ccnc21

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.36
ADRA2C P18825 1/20 0.36
ALDH1A1 P00352 3/20 0.34
ADRA1A P35348 3/20 0.33
MAPT P10636 2/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
TSHR P16473 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ADRA1D P25100 2/20 0.33
ADRA1B P35368 2/20 0.33
HTR1A P08908 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4784878 0.85 NISCH (0.33) TSHR
SCHEMBL14160384 0.81 KDM4E (0.45) ADRA2CALDH1A1ADRA1AKDM4EADRA1D
SCHEMBL4782058 0.75 ADRA2C (0.57) HTR2CADRA2CALDH1A1MAPTKDM4E
SCHEMBL4780757 0.75 HTR2C (0.36) HTR2CADRA2CALDH1A1MAPTKDM4E
Hydrochloric Acid SCHEMBL4780986 0.74 ADRA2C (0.56) HTR2CADRA2CALDH1A1MAPTKDM4E
SCHEMBL3954178 0.73 ADRA2C (0.40) ADRA2CADRA1AKDM4EADRA1DADRA1B
SCHEMBL1267500 0.68 ALDH1A1 (0.62) HTR2CADRA2CALDH1A1MAPTKDM4E
SCHEMBL929673 0.65 TACR3 (0.37) ALDH1A1KDM4E
SCHEMBL13170398 0.65 HTR2C (0.50) HTR2CALDH1A1
SCHEMBL22776034 0.64 KDM4E (0.46) ALDH1A1ADRA1AMAPTTSHRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed