SCHEMBL4802544

SCHEMBL4802544

CC(=O)Nc1ccccc1OCC(O)CN1CCC(n2c(=O)[nH]c3ccccc32)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 10/20 0.66
OPRM1 P35372 8/20 0.57
PLD1 Q13393 2/20 0.53
PLD2 O14939 1/20 0.53
ADRA1D P25100 2/20 0.53
ADRA1A P35348 2/20 0.53
ADRA1B P35368 2/20 0.53
ADRB2 P07550 1/20 0.53
ADRB1 P08588 1/20 0.53
ADRB3 P13945 1/20 0.53
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
PMP22 Q01453 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ABCB11 O95342 1/20 0.49
CHRM1 P11229 1/20 0.48
DRD2 P14416 1/20 0.48
KCNH2 Q12809 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4798788 0.99 OPRL1 (0.65) OPRL1OPRM1PLD1PLD2ADRA1D
SCHEMBL11648606 0.92 OPRL1 (0.63) OPRL1OPRM1PLD1PLD2ADRA1D
SCHEMBL4808944 0.91 OPRL1 (0.57) OPRL1OPRM1PLD1PLD2CHRM1
SCHEMBL4808096 0.90 OPRL1 (0.60) OPRL1OPRM1PLD1PLD2ABCB11
Hydrochloric Acid SCHEMBL4805718 0.90 OPRL1 (0.56) OPRL1OPRM1PLD1PLD2ADRA1D
SCHEMBL6628494 0.90 OPRL1 (0.60) OPRL1OPRM1PLD1PLD2ABCB11
Hydrochloric Acid SCHEMBL4805706 0.90 OPRL1 (0.56) OPRL1OPRM1PLD1PLD2ADRA1D
SCHEMBL6628489 0.90 OPRL1 (0.60) OPRL1OPRM1PLD1PLD2ABCB11
Hydrochloric Acid SCHEMBL4806574 0.89 OPRL1 (0.61) OPRL1OPRM1PLD1PLD2ADRA1D
SCHEMBL4807271 0.89 OPRL1 (0.67) OPRL1OPRM1PLD1PLD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116435-A1 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2004-06-17 US claimed
WO-2002074763-A9 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS ASTRAZENECA AB (SE) 2002-10-24 WO claimed
US-7388020-B2 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2008-06-17 US disclosed
US-20040116435-A1 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2004-06-17 US disclosed
EP-1373248-A1 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS AstraZeneca AB (SE) 2004-01-02 EP disclosed
WO-2002074763-A1 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS ASTRAZENECA AB (SE) 2002-09-26 WO disclosed