SCHEMBL6628489

SCHEMBL6628489

CC(=O)Nc1ccccc1OC[C@@H](O)CN1CCC(n2c(=O)[nH]c3cc(Cl)ccc32)CC1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 2/20 0.60
PLD1 Q13393 11/20 0.56
PLD2 O14939 10/20 0.56
CCR1 P32246 1/20 0.54
ABCB11 O95342 1/20 0.53
DRD2 P14416 2/20 0.51
HTR1A P08908 1/20 0.51
ADRA2A P08913 1/20 0.51
HTR2A P28223 1/20 0.51
SLC6A4 P31645 1/20 0.51
DRD3 P35462 1/20 0.51
OPRM1 P35372 1/20 0.51
CHRM1 P11229 2/20 0.50
YEATS4 O95619 1/20 0.50
MLLT3 P42568 1/20 0.50
MLLT1 Q03111 1/20 0.50
KCNH2 Q12809 1/20 0.50
YEATS2 Q9ULM3 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6628494 1.00 OPRL1 (0.60) OPRL1PLD1PLD2CCR1ABCB11
Trifluoroacetic Acid SCHEMBL4799510 0.95 OPRL1 (0.55) OPRL1PLD1PLD2CCR1ABCB11
SCHEMBL4808096 0.94 OPRL1 (0.60) OPRL1PLD1PLD2CCR1ABCB11
SCHEMBL4850139 0.92 PLD1 (0.59) OPRL1PLD1PLD2CCR1DRD2
SCHEMBL4808944 0.91 OPRL1 (0.57) OPRL1PLD1PLD2CCR1DRD2
Hydrochloric Acid SCHEMBL4805718 0.91 OPRL1 (0.56) OPRL1PLD1PLD2CCR1DRD2
Hydrochloric Acid SCHEMBL4805706 0.91 OPRL1 (0.56) OPRL1PLD1PLD2CCR1DRD2
SCHEMBL4802544 0.90 OPRL1 (0.66) OPRL1PLD1PLD2ABCB11DRD2
SCHEMBL4807137 0.90 PLD1 (0.59) OPRL1PLD1PLD2CCR1DRD2
Hydrochloric Acid SCHEMBL4798788 0.90 OPRL1 (0.65) OPRL1PLD1PLD2ABCB11DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116435-A1 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2004-06-17 US claimed
EP-1373248-A1 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS AstraZeneca AB (SE) 2004-01-02 EP disclosed
WO-2002074763-A9 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS ASTRAZENECA AB (SE) 2002-10-24 WO disclosed
WO-2002074763-A1 BENZIMIDAZOL DERIVATIVES MODULATE CHEMOKINE RECEPTORS ASTRAZENECA AB (SE) 2002-09-26 WO disclosed