Guaiacol

Guaiacol

SCHEMBL480341

CCCCCCOc1c(O)cccc1CC.COc1ccccc1O.c1cnnnc1

nearest known ligand 0.44

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.42
PTGS2 P35354 1/20 0.42
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
PPARA Q07869 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
TP53 P04637 1/20 0.40
TSHR P16473 1/20 0.40
CYP3A4 P08684 2/20 0.38
MEN1 O00255 1/20 0.38
NR1I2 O75469 1/20 0.38
LMNA P02545 1/20 0.38
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
MAPT P10636 1/20 0.38
OPRK1 P41145 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Guaiacol SCHEMBL3387344 1.00 ALOX5 (0.42) ALOX5PTGS2CNR1CNR2PPARA
Guaiacol SCHEMBL3959515 0.92 ALOX5 (0.49) ALOX5PTGS2CNR1CNR2PPARA
SCHEMBL29286378 0.91 BID (0.42) PPARAMEN1MAPTKMT2A
Guaiacol SCHEMBL5320834 0.90 CNR1 (0.43) ALOX5PTGS2CNR1CNR2CA1
Anisole SCHEMBL27966148 0.89 MAPT (0.39) PPARAMAPT
Guaiacol SCHEMBL268884 0.88 CNR1 (0.40) ALOX5CNR1CNR2CA1CA2
Guaiacol SCHEMBL5483774 0.86 CA1 (0.49) ALOX5PTGS2CNR1CNR2CA1
Guaiacol SCHEMBL5320116 0.86 CA1 (0.49) ALOX5PTGS2CNR1CNR2CA1
SCHEMBL790778 0.85 ELANE (0.38) ALOX5PTGS2CNR1CNR2PPARA
SCHEMBL15162949 0.85 ELANE (0.38) ALOX5PTGS2CNR1CNR2PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 80 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2916814-A1 COMPOSITION CONTAINING A CELLULOSE DERIVED CAPSULE WITH A SUNSCREEN Colabs International Corporation (US) 2015-09-16 EP claimed
WO-2014074555-A1 COMPOSITION CONTAINING A CELLULOSE DERIVED CAPSULE WITH A SUNSCREEN CoLabs International Corporation (US) 2014-05-15 WO claimed
JP-4664289-B2 2011-04-06 JP claimed
EP-1337145-A4 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PROD INC (US) 2009-05-27 EP claimed
EP-2061308-A2 A WATER BASED CLEAR SUNSCREEN AND INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2009-05-27 EP claimed
EP-1784158-A4 IMPROVED TOPICAL SKIN CARE COMPOSITIONS AVON PROD INC (US) 2009-03-11 EP claimed
WO-2008024738-A2 A WATER BASED CLEAR SUNSCREEN AND INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2008-02-28 WO claimed
EP-1648853-A4 COMPOSITIONS CONTAINING PHENETHYL ARYL ESTERS AS SOLUBILIZING AGENTS FOR ACTIVE ORGANIC COMPOUNDS ISP INVESTMENTS INC (US) 2008-01-02 EP claimed
JP-2007518689-A 2007-07-12 JP claimed
EP-1784158-A1 IMPROVED TOPICAL SKIN CARE COMPOSITIONS AVON PRODUCTS, INC. (US) 2007-05-16 EP claimed
EP-1648853-A2 COMPOSITIONS CONTAINING PHENETHYL ARYL ESTERS AS SOLUBILIZING AGENTS FOR ACTIVE ORGANIC COMPOUNDS Bertz, Steven H. (US) 2006-04-26 EP claimed
WO-2006026168-A1 IMPROVED TOPICAL SKIN CARE COMPOSITIONS AVON PRODUCTS, INC. (US) 2006-03-09 WO claimed
WO-2005065136-A2 OIL IN SILICONE EMULSIONS AND COMPOSITIONS CONTAINING SAME AVON PRODUCTS, INC. (US) 2005-07-21 WO claimed
WO-2005065154-A2 NOVEL ESTERS OF ARYL BENZIMIDAZOLE SULFONIC ACIDS AND SUNSCREEN COMPOSITIONS CONTAINING SAME AVON PRODUCTS, INC. (US) 2005-07-21 WO claimed
WO-2005009341-A2 COMPOSITIONS CONTAINING PHENETHYL ARYL ESTERS AS SOLUBILIZING AGENTS FOR ACTIVE ORGANIC COMPOUNDS ISP INVESTMENTS INC. (US) 2005-02-03 WO claimed
EP-1337145-A1 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2003-08-27 EP claimed
WO-2003051279-A2 TOPICAL COMPOSITIONS AND METHODS OF APPLICATION AVON PRODUCTS, INC. (US) 2003-06-26 WO claimed
WO-2002043656-A2 WATER-IN-OIL INSECT REPELLENT COMPOSITION AND METHOD OF APPLICATION TO THE SKIN AVON PRODUCTS, INC. (US) 2002-06-06 WO claimed
WO-2002043489-A1 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2002-06-06 WO claimed
WO-2024137719-A1 SPRAYABLE SUNSCREEN COMPOSITIONS CONTAING OIL-IN-WATER EMULSIONS CONTAINING SUBMICRON HYDROPHOBIC AGENTS AND METHODS OF USE THEREOF Leading Edge Innovations, LLC (US) 2024-06-27 WO disclosed
WO-2024137566-A1 SPRAYABLE SUNSCREEN COMPOSITIONS CONTAINING OIL-IN-WATER DISPERSIONS OF HYDROPHOBIC AGENTS AND POLYMER OR COPOLYMER FRAGMENTS, OR COMBINATIONS THEREOF, AND METHODS OF USE THEREOF Leading Edge Innovations, LLC (US) 2024-06-27 WO disclosed
WO-2018109469-A1 NOVEL PROCESS ITACONIX (U.K.) LIMITED (GB) 2018-06-21 WO disclosed
EP-3313534-A1 SUPERABSORBENT POLYMERS AND STARCH POWDERS FOR USE IN SKIN CARE COMPOSITIONS The Procter and Gamble Company (US) 2018-05-02 EP disclosed
EP-3288528-A1 SILK-BASED MOISTURIZER COMPOSITIONS AND METHODS THEREOF Silk Therapeutics Inc. (US) 2018-03-07 EP disclosed
EP-3280498-A1 PROTECTIVE ACTION OF LUTEIN AGAINST BLUE LIGHT ON HUMAN SKIN CELL LINES Kemin Industries, Inc. (US) 2018-02-14 EP disclosed
EP-3191074-A1 COSMETIC COMPOSITIONS AND METHODS FOR INHIBITING MELANIN SYNTHESIS The Procter and Gamble Company (US) 2017-07-19 EP disclosed
EP-3122428-A1 SPRAYABLE SUNSCREEN COMPOSITIONS AND METHODS Inolex Investment Corporation (US) 2017-02-01 EP disclosed
WO-2017004108-A1 SUPERABSORBENT POLYMERS AND STARCH POWDERS FOR USE IN SKIN CARE COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 2017-01-05 WO disclosed
WO-2016176633-A1 SILK-BASED MOISTURIZER COMPOSITIONS AND METHODS THEREOF Silk Therapeutics, Inc. (US) 2016-11-03 WO disclosed
WO-2016164744-A1 PROTECTIVE ACTION OF LUTEIN AGAINST BLUE LIGHT ON HUMAN SKIN CELL LINES KEMIN INDUSTRIES, INC. (US) 2016-10-13 WO disclosed
WO-2016040757-A1 COSMETIC COMPOSITIONS AND METHODS FOR INHIBITING MELANIN SYNTHESIS THE PROCTER & GAMBLE COMPANY (US) 2016-03-17 WO disclosed
WO-2016032852-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF PHOTOAGING AND OTHER SKIN CONDITIONS PRO TRANSIT NANOTHERAPY LLC (US) 2016-03-03 WO disclosed
WO-2015148999-A1 SPRAYABLE SUNSCREEN COMPOSITIONS AND METHODS INOLEX INVESTMENT CORPORATION (US) 2015-10-01 WO disclosed
EP-2919748-A1 COSMETIC COMPOSITIONS AND METHODS FOR INHIBITING MELANIN SYNTHESIS The Procter & Gamble Company (US) 2015-09-23 EP disclosed
EP-2916814-A1 COMPOSITION CONTAINING A CELLULOSE DERIVED CAPSULE WITH A SUNSCREEN Colabs International Corporation (US) 2015-09-16 EP disclosed
CN-104718273-A Compositions, apparatus, systems, and methods for resolving electronic excited states HALLSTAR INNOVATIONS CORP 2015-06-17 CN disclosed
WO-2014179520-A1 COSMETIC COMPOSITIONS AND METHODS FOR INHIBITING MELANIN SYNTHESIS THE PROCTER & GAMBLE COMPANY (US) 2014-11-06 WO disclosed
EP-2755625-A1 SHELLAC BASED SPRAYABLE SUNSCREEN Mantrose-Haeuser Co. Inc. (US) 2014-07-23 EP disclosed
WO-2014074555-A1 COMPOSITION CONTAINING A CELLULOSE DERIVED CAPSULE WITH A SUNSCREEN CoLabs International Corporation (US) 2014-05-15 WO disclosed
WO-2013039826-A1 SHELLAC BASED SPRAYABLE SUNSCREEN MANTROSE-HAEUSER CO., INC. (US) 2013-03-21 WO disclosed
EP-2558059-A2 COMPOSITIONS AND METHODS FOR SPF ENHANCEMENT BY HIGH CONCENTRATION COSMETIC POWDER FORMULATIONS U.S. Cosmetics Corporation (US) 2013-02-20 EP disclosed
CN-101802097-B Phosphoric acid esters containing phosphorus atoms bridged by diol units CLARIANT FINANCE BVI LTD 2012-11-14 CN disclosed
CN-1871203-B Composition comprising phenethyl aryl esters as solubilizers for active organic compounds ISP INVESTMENTS INC 2012-11-14 CN disclosed
CN-101802096-B Aqueous compositions containing alkoxylated phosphoric triesters CLARIANT FINANCE BVI LTD 2012-07-18 CN disclosed
EP-2414408-A1 CATIONIC COMB COPOLYMERS, PREPARATION THEREOF AND USE THEREOF IN COSMETIC, PHARMACEUTICAL AND DERMATOLOGICAL FORMULATIONS Clariant Finance (BVI) Limited (VG) 2012-02-08 EP disclosed
EP-2411427-A1 POLYMERS BASED ON ACRYLIC, METHACRYLIC OR ETHACRYLIC AMIDOALKYL SULFONIC ACID OR SALTS AND CARBOXYALKYL ACRYLATE, METHACRYLATE OR ETHACRYLATE OR OLIGOMERS OF SAID CARBOXY COMPOUNDS Clariant Finance (BVI) Limited (VG) 2012-02-01 EP disclosed
WO-2011130358-A2 COMPOSITIONS AND METHODS FOR SPF ENHANCEMENT BY HIGH CONCENTRATION COSMETIC POWDER FORMULATIONS U.S. COSMETICS CORPORATION (US) 2011-10-20 WO disclosed
WO-2011119592-A1 PLANT EXTRACTS, COMPOSITIONS CONTAINING SAME, AND USES THEREOF DEO NAMITA (US) 2011-09-29 WO disclosed
EP-2274057-A1 SUNSCREENS DSM IP Assets B.V. (NL) 2011-01-19 EP disclosed
WO-2010112185-A1 CATIONIC COMB COPOLYMERS, PREPARATION THEREOF AND USE THEREOF IN COSMETIC, PHARMACEUTICAL AND DERMATOLOGICAL FORMULATIONS CLARIANT INTERNATIONAL LTD (CH) 2010-10-07 WO disclosed
WO-2010108634-A1 POLYMERS BASED ON ACRYLIC, METHACRYLIC OR ETHACRYLIC AMIDOALKYL SULFONIC ACID OR SALTS AND CARBOXYALKYL ACRYLATE, METHACRYLATE OR ETHACRYLATE OR OLIGOMERS OF SAID CARBOXY COMPOUNDS CLARIANT INTERNATIONAL LTD (CH) 2010-09-30 WO disclosed
WO-2010100032-A1 A SKIN COLOUR SHADE CARD UNILEVER NV (NL) 2010-09-10 WO disclosed
EP-2176350-A2 AQUEOUS COMPOSITIONS CONTAINING ALKOXYLATED PHOSPHORIC ACID TRIESTERS Clariant Finance (BVI) Limited (VG) 2010-04-21 EP disclosed
WO-2009138485-A1 SUNSCREENS DSM IP ASSETS B.V. (NL) 2009-11-19 WO disclosed
EP-1802290-A4 SOLUBILIZING AGENTS FOR ACTIVE OR FUNCTIONAL ORGANIC COMPOUNDS ISP INVESTIMENTS INC (US) 2009-08-19 EP disclosed
EP-1337145-A4 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PROD INC (US) 2009-05-27 EP disclosed
EP-2061308-A2 A WATER BASED CLEAR SUNSCREEN AND INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2009-05-27 EP disclosed
WO-2009020518-A1 TOPICAL ACNE VULGARIS COMPOSITION WITH A SUNSCREEN DOW PHARMACEUTICAL SCIENCES (US) 2009-02-12 WO disclosed
WO-2009015857-A2 AQUEOUS COMPOSITIONS CONTAINING ALKOXYLATED PHOSPHORIC ACID TRIESTERS CLARIANT INTERNATIONAL LTD (CH) 2009-02-05 WO disclosed
EP-1910271-A4 SUNLESS TANNING SUBSTRATE PLAYTEX PRODUCTS INC (US) 2008-11-19 EP disclosed
EP-1910271-A2 SUNLESS TANNING SUBSTRATE PLAYTEX PRODUCTS, INC. (US) 2008-04-16 EP disclosed
WO-2008024738-A2 A WATER BASED CLEAR SUNSCREEN AND INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2008-02-28 WO disclosed
WO-2008016837-A2 AQUEOUS COMPOSITIONS CONTAINING A HYDROPHOBIC MATERIAL ISP INVESTMENTS INC. (US) 2008-02-07 WO disclosed
WO-2008002609-A2 HYDROQUINONE COMPOSITIONS FOR SKIN LIGHTENING APPLIED GENETICS INCORPORATED DERMATICS (US) 2008-01-03 WO disclosed
EP-1827111-A2 METHOD AND COMPOSITION FOR REDUCING THE APPEARANCE OF WRINKLES AVON PRODUCTS, INC. (US) 2007-09-05 EP disclosed
EP-1802290-A2 SOLUBILIZING AGENTS FOR ACTIVE OR FUNCTIONAL ORGANIC COMPOUNDS ISP Investiments Inc. (US) 2007-07-04 EP disclosed
CN-1305765-C Process for preparation of aqueous suspensions of anionic colloidal silica having a neutral phand applications thereof CLARIANT INT LTD (US) 2007-03-21 CN disclosed
WO-2007005740-A2 SUNLESS TANNING SUBSTRATE PLAYTEX PRODUCTS, INC. (US) 2007-01-11 WO disclosed
WO-2006069072-A2 METHOD AND COMPOSITION FOR REDUCING THE APPEARANCE OF WRINKLES AVON PRODUCTS INC. (US) 2006-06-29 WO disclosed
WO-2006041506-A2 SOLUBILIZING AGENTS FOR ACTIVE OR FUNCTIONAL ORGANIC COMPOUNDS ISP INVESTMENTS INC. (US) 2006-04-20 WO disclosed
WO-2005065136-A2 OIL IN SILICONE EMULSIONS AND COMPOSITIONS CONTAINING SAME AVON PRODUCTS, INC. (US) 2005-07-21 WO disclosed
WO-2005065154-A2 NOVEL ESTERS OF ARYL BENZIMIDAZOLE SULFONIC ACIDS AND SUNSCREEN COMPOSITIONS CONTAINING SAME AVON PRODUCTS, INC. (US) 2005-07-21 WO disclosed
WO-2005062860-A2 NEW SUNSCREEN COMPOUNDS AND COMPOSITIONS CONTAINING SAME AND METHODS FOR USE THEREOF AVON PRODUCTS, INC. (US) 2005-07-14 WO disclosed
EP-1490018-A2 SUNSCREEN COMPOSITIONS AND METHODS AND MATERIALS FOR PRODUCING THE SAME The C.P. Hall Company (US) 2004-12-29 EP disclosed
CN-1484614-A Process for preparation of aqueous suspensions of anionic colloidal silica having a neutral phand applications thereof 克莱里安特财务(BVI)有限公司 2004-03-24 CN disclosed
WO-2003075878-A2 METHODS OF MAKING AND SELLING A SUNSCREEN COMPOSITION THE C.P. HALL COMPANY (US) 2003-09-18 WO disclosed
WO-2003075877-A2 SUNSCREEN COMPOSITIONS AS WELL AS METHODS AND MATERIALS FOR PRODUCING THE SAME, WHEREIN THE PHOTODECAY RATE OF THE FILTER SYSTEM IS REDUCED BY CONTROLLING THE POLARITY OF THE SOLVENT SYSTEM THE C.P. HALL COMPANY (US) 2003-09-18 WO disclosed
EP-1337145-A1 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2003-08-27 EP disclosed
WO-2003051279-A2 TOPICAL COMPOSITIONS AND METHODS OF APPLICATION AVON PRODUCTS, INC. (US) 2003-06-26 WO disclosed
WO-2002043489-A1 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2002-06-06 WO disclosed
WO-2002043489-A1 ANHYDROUS INSECT REPELLENT COMPOSITION AVON PRODUCTS, INC. (US) 2002-06-06 WO disclosed