SCHEMBL4806014

SCHEMBL4806014

CC(C)(C)c1csc(N(N)C(=O)c2ccc(Cl)cc2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.52
KDM4E B2RXH2 5/20 0.52
TDP1 Q9NUW8 1/20 0.52
GRM1 Q13255 2/20 0.45
FFAR2 O15552 1/20 0.43
RAB9A P51151 4/20 0.41
CFTR P13569 1/20 0.41
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HTT P42858 2/20 0.38
MAPK1 P28482 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
GAA P10253 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4797120 0.75 GRM1 (0.59) NPC1KDM4EGRM1RAB9AMAPT
SCHEMBL4798879 0.73 NPC1 (0.59) NPC1KDM4EGRM1RAB9AMAPT
SCHEMBL20791859 0.70 NPC1 (0.76) NPC1KDM4ETDP1FFAR2RAB9A
SCHEMBL3345136 0.69 MAPT (0.50) NPC1KDM4ETDP1GRM1RAB9A
SCHEMBL3340907 0.68 KDM4E (1.00) NPC1KDM4ETDP1FFAR2RAB9A
SCHEMBL10931661 0.68 UCHL1 (0.49) NPC1KDM4ETDP1GRM1RAB9A
SCHEMBL8167107 0.67 CES2 (0.45) NPC1KDM4ERAB9AMAPTSMN1; SMN2
Hydrochloric Acid SCHEMBL11830537 0.65 TP53 (0.56) NPC1KDM4ETDP1RAB9AMAPT
SCHEMBL4798176 0.65 GRM1 (0.55) NPC1KDM4EGRM1RAB9AMAPT
SCHEMBL10591755 0.64 ELANE (0.42) NPC1KDM4ETDP1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008052804-A1 THIAZOLHYDRAZIDES FOR TREATMENT OF NEURODEGENERATIVE DISEASES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2008-05-08 WO disclosed