SCHEMBL4806170

SCHEMBL4806170

Cn1c(Cc2ccc(Br)c(Oc3cc(C#N)cc(C#N)c3)c2F)n[nH]c1=O

nearest known ligand 0.70

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.70
KCNH2 Q12809 4/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
MTNR1B P49286 1/20 0.38
EPAS1 Q99814 4/20 0.31
VEGFA P15692 1/20 0.31
MAPK1 P28482 1/20 0.31
APOBEC3G Q9HC16 1/20 0.31
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4801545 0.93 CYP3A4 (0.82) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4807848 0.92 CYP3A4 (0.63) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4808072 0.90 CYP3A4 (0.73) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4805825 0.89 CYP3A4 (0.87) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4800446 0.88 CYP3A4 (0.76) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL3664378 0.86 CYP3A4 (0.71) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4807889 0.83 CYP3A4 (0.84) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4808573 0.83 CYP3A4 (0.84) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL14262139 0.83 CYP3A4 (1.00) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B
SCHEMBL4580827 0.82 CYP3A4 (0.54) CYP3A4KCNH2CYP2C9CYP2C19MTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348345-B2 Nonnucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2008-03-25 US disclosed
US-20070179157-A1 Nonnucleoside reverse transcriptase inhibitors DUNN JAMES P 2007-08-02 US disclosed
US-7208509-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-04-24 US disclosed
US-7208509-B2 Non-nucleoside reverse transcriptase inhibitors ROCHE PALO ALTO LLC (US) 2007-04-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070179157-A1 Nonnucleoside reverse transcriptase inhibitors RRM2, RRM2B, SAMHD1 CYP3A4 438/4885KCNH2 3216/4885CYP2C9 1755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.