SCHEMBL4806633

SCHEMBL4806633

O=C(Nc1ccccc1OCC(O)CN1CCC(n2c(=O)oc3ccccc32)CC1)c1ccc(Cl)cc1

nearest known ligand 0.66

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 5/20 0.66
SCN5A Q14524 5/20 0.66
SCN9A Q15858 5/20 0.66
PLD1 Q13393 3/20 0.55
ABCB11 O95342 1/20 0.45
CCR1 P32246 4/20 0.44
KCNH2 Q12809 1/20 0.44
HRH1 P35367 1/20 0.44
CCR3 P51677 1/20 0.44
OPRL1 P41146 2/20 0.43
HSD11B1 P28845 1/20 0.42
DRD4 P21917 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
CYP2D6 P10635 2/20 0.41
PLD2 O14939 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4800626 0.94 SCN1A (0.75) SCN1ASCN5ASCN9APLD1CCR1
SCHEMBL4803367 0.92 SCN1A (0.66) SCN1ASCN5ASCN9APLD1CCR1
SCHEMBL4800272 0.87 SCN1A (0.69) SCN1ASCN5ASCN9APLD1ABCB11
Hydrochloric Acid SCHEMBL4808473 0.86 SCN1A (0.68) SCN1ASCN5ASCN9APLD1ABCB11
SCHEMBL4806019 0.84 OPRL1 (0.63) PLD1KCNH2OPRL1PLD2
SCHEMBL4799829 0.81 OPRL1 (0.57) PLD1CCR1KCNH2HRH1CCR3
SCHEMBL4807512 0.80 PLD2 (0.66) PLD1KCNH2OPRL1PLD2
SCHEMBL4803925 0.78 PLD2 (0.55) PLD1KCNH2OPRL1PLD2
SCHEMBL4806618 0.78 OPRL1 (0.62) PLD1OPRL1PLD2
Hydrochloric Acid SCHEMBL4806574 0.77 OPRL1 (0.61) SCN1ASCN5ASCN9APLD1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7388020-B2 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2008-06-17 US claimed
US-20040116435-A1 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2004-06-17 US claimed
US-7388020-B2 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2008-06-17 US disclosed
US-20040116435-A1 Benzimidazol derivatives modulate chemokine receptors ASTRAZENECA AB (SE) 2004-06-17 US disclosed