SCHEMBL480738

SCHEMBL480738

C=C(CCc1ccc(-c2ccccc2)cc1)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 4/20 0.67
MMP12 P39900 5/20 0.59
NAAA Q02083 1/20 0.53
FFAR4 Q5NUL3 1/20 0.51
HDAC2 Q92769 2/20 0.50
ABCC4 O15439 1/20 0.50
LMNA P02545 1/20 0.50
GAA P10253 1/20 0.50
TSHR P16473 1/20 0.50
PTGS1 P23219 1/20 0.50
HTT P42858 1/20 0.50
CES1 P23141 2/20 0.49
HDAC1 Q13547 1/20 0.49
MMP13 P45452 4/20 0.49
KEAP1 Q14145 1/20 0.48
CNR2 P34972 1/20 0.48
MMP2 P08253 1/20 0.47
MMP9 P14780 1/20 0.47
MMP14 P50281 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1920267 0.89 FFAR1 (0.58) FFAR1MMP12NAAAHDAC2ABCC4
SCHEMBL17940817 0.89 FFAR1 (0.64) FFAR1FFAR4HDAC2HTTHDAC1
SCHEMBL30529 0.88 KEAP1 (0.61) FFAR1HDAC2HTTHDAC1KEAP1
SCHEMBL17940796 0.86 FFAR1 (0.50) FFAR1MMP12FFAR4HDAC2
SCHEMBL17940809 0.86 FFAR1 (0.49) FFAR1MMP12NAAAFFAR4HDAC2
SCHEMBL1920994 0.85 FFAR1 (0.55) FFAR1FFAR4HDAC2LMNAHTT
SCHEMBL1920986 0.84 FFAR1 (0.50) FFAR1MMP12FFAR4KEAP1
Succinic Acid SCHEMBL14801749 0.83 KEAP1 (0.67) FFAR1FFAR4HDAC2HDAC1KEAP1
SCHEMBL17940826 0.82 SRD5A2 (0.54) FFAR1LMNAHTTHDAC1KEAP1
SCHEMBL17940829 0.82 F2RL1 (0.57) FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 45 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4121802-B1 HIGH REFRACTIVE INDEX SILOXANE INSERT MATERIALS FOR EMBEDDED CONTACT LENSES ALCON INC (CH) 2024-07-17 EP claimed
EP-3728339-B1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS AMO Ireland (IE) 2022-07-06 EP claimed
EP-2303331-B1 OPHTHALMIC DEVICE HAVING THERAPEUTIC AGENT DELIVERY CAPABILITY AND METHOD OF FORMING SAME ALCON INC (CH) 2022-01-26 EP claimed
EP-3200840-B1 LOW-WATER CONTENT ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES ALCON INC (CH) 2021-11-17 EP claimed
US-10920000-B2 Light diffusing agent, light diffusing resin composition and molded body MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) 2021-02-16 US claimed
EP-3200839-B1 HYDROPHOBIC ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES NOVARTIS AG (CH) 2019-09-04 EP claimed
EP-3223870-B1 WET-PACK INTRAOCULAR LENS MATERIALS WITH HIGH REFRACTIVE INDEX NOVARTIS AG (CH) 2018-09-26 EP claimed
EP-3077016-B1 SOFT ACRYLIC MATERIALS WITH HIGH REFRACTIVE INDEX AND MINIMIZED GLISTENING NOVARTIS AG (CH) 2018-05-16 EP claimed
EP-2906970-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS WITH REDUCED TACK NOVARTIS AG (CH) 2016-11-23 EP claimed
EP-2684903-B1 RADICAL POLYMERIZABLE COMPOSITION, HARDENED PRODUCT THEREOF, AND PLASTIC LENS THEREOF DAINIPPON INK & CHEMICALS (JP) 2015-12-16 EP claimed
US-9156931-B2 Radical polymerizable composition, cured product, and plastic lens DIC CORPORATION (JP) 2015-10-13 US claimed
EP-2664635-B1 RADICALLY POLYMERIZABLE COMPOSITION, CURED PRODUCT, AND PLASTIC LENS DAINIPPON INK & CHEMICALS (JP) 2015-05-20 EP claimed
EP-2586802-B1 RADICALLY POLYMERIZABLE COMPOSITION, CURED PRODUCT AND PLASTIC LENS DAINIPPON INK & CHEMICALS (JP) 2014-12-24 EP claimed
EP-2582409-B1 HIGH REFRACTIVE INDEX, ACRYLIC OPHTHALMIC DEVICE MATERIALS WITH REDUCED GLISTENINGS NOVARTIS AG (CH) 2014-09-10 EP claimed
US-20140148525-A1 RADICAL POLYMERIZABLE COMPOSITION, CURED PRODUCT, AND PLASTIC LENS DIC CORPORATION (JP) 2014-05-29 US claimed
EP-2225325-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS ALCON INC (CH) 2011-06-01 EP claimed
EP-1080382-B1 HIGH REFRACTIVE INDEX OPHTHALMIC DEVICE MATERIALS ALCON INC (CH) 2009-07-08 EP claimed
EP-3728339-B1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS AMO Ireland (IE) 2022-07-06 EP disclosed
US-20100304153-A1 SURFACE-TREATED RESIN, METHOD FOR PRODUCING THE SAME, AND USE OF THE SAME OMRON CORPORATION (JP) 2010-12-02 US disclosed
EP-2082872-A1 SURFACE-TREATED RESIN, METHOD FOR PRODUCING THE SAME, AND USE OF THE SAME OMRON Corporation, a corporation of Japan (JP) 2009-07-29 EP disclosed