SCHEMBL4809982

SCHEMBL4809982

CCCCCc1nc(C)sc1C(=O)OCC

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
CYP1A2 P05177 1/20 0.48
NPC1 O15118 1/20 0.47
TSHR P16473 2/20 0.45
HPGD P15428 2/20 0.44
HSD17B10 Q99714 3/20 0.44
GAA P10253 1/20 0.44
HTT P42858 1/20 0.44
CDC7 O00311 6/20 0.42
DBF4 Q9UBU7 6/20 0.42
LMNA P02545 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CYP2C9 P11712 1/20 0.40
MAPT P10636 1/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7613881 0.89 ALDH1A1 (0.51) ALDH1A1CYP1A2NPC1TSHRHPGD
SCHEMBL1919240 0.87 ALDH1A1 (0.47) ALDH1A1CYP1A2TSHRHPGDHSD17B10
SCHEMBL9644349 0.83 GPR35 (0.44) ALDH1A1TSHRHPGDHTTNPSR1
SCHEMBL21771163 0.82 NPC1 (0.52) ALDH1A1CYP1A2NPC1TSHRHPGD
SCHEMBL2823884 0.82 ALDH1A1 (0.63) ALDH1A1CYP1A2NPC1TSHRHPGD
SCHEMBL2823911 0.82 ALDH1A1 (0.48) ALDH1A1CYP1A2TSHRHPGDHSD17B10
SCHEMBL9644203 0.81 GPR35 (0.47) ALDH1A1HTTNPSR1MAPT
SCHEMBL2719635 0.81 NPC1 (0.49) ALDH1A1CYP1A2NPC1TSHRHPGD
SCHEMBL12324407 0.80 NPC1 (0.50) ALDH1A1CYP1A2NPC1TSHRHPGD
SCHEMBL11156431 0.80 ALDH1A1 (0.50) ALDH1A1CYP1A2NPC1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008087611-A2 PYRROLIDINE- AND PIPERIDINE- BIS-AMIDE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-07-24 WO disclosed