SCHEMBL4812600

SCHEMBL4812600

Cc1cccc(C)c1OC(=O)Cl

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 2/20 0.48
HPGD P15428 2/20 0.48
HSD17B10 Q99714 2/20 0.48
KMT2A Q03164 5/20 0.45
MEN1 O00255 3/20 0.45
ATM Q13315 1/20 0.45
PTPN1 P18031 1/20 0.42
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11611613 0.83 TSHR (0.48) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL8764787 0.81 L3MBTL1 (0.55) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL2059537 0.79 KDM4E (0.71) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL982574 0.79 L3MBTL1 (0.58) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL6771381 0.78 L3MBTL1 (0.45) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL2948942 0.77 KDM4E (0.42) ALDH1A1KDM4EKMT2AMEN1ATM
SCHEMBL10959076 0.77 L3MBTL1 (0.52) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL10523979 0.77 L3MBTL1 (0.52) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL20921192 0.77 TSHR (0.43) L3MBTL1SMN1; SMN2ALDH1A1KDM4EHPGD
SCHEMBL8463126 0.77 POLB (0.56) L3MBTL1ALDH1A1KMT2AMEN1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108530297-B Preparation method of 2-chloro-3-methylbenzoic acid and intermediate thereof 联化科技股份有限公司 2021-09-24 CN claimed
EP-1622910-A1 FUSED PYRIMIDINE DERIVATIVES WITH CRF ACTIVITY F. HOFFMANN-LA ROCHE AG (CH) 2006-02-08 EP claimed
WO-2004099209-A1 FUSED PYRIMIDINE DERIVATIVES WITH CRF ACTIVITY F. HOFFMANN-LA-ROCHE AG (CH) 2004-11-18 WO claimed
US-5874655-A Process for the preparation of chlorinated aromatics BAYER AKTIENGESELLSCHAFT (DE) 1999-02-23 US claimed
EP-0694513-B1 Process for preparing chlorinated aromatic compounds BAYER AG (DE) 1998-10-28 EP claimed
EP-0590259-B1 Process for the preparation of halogenated aromatic compounds BAYER AG (DE) 1997-10-29 EP claimed
US-5306849-A Process for the preparation of halogenated aromatics BAYER AKTIENGESELLSCHAFT (DE) 1994-04-26 US claimed
JP-7304697-A None JP disclosed
US-20200338087-A9 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-10-29 US disclosed
US-20200338087-A9 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-10-29 US disclosed
US-20190343842-A1 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-11-14 US disclosed
US-20190343842-A1 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS DANA-FARBER CANCER INSTITUTE, INC. (US) 2019-11-14 US disclosed
EP-3536323-A1 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS Dana Farber Cancer Institute, Inc. (US) 2019-09-11 EP disclosed
US-4983616-A Analgesics, cognition activators HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-01-08 US disclosed
US-4751173-A USING QUATERNARY COMPOUND; RAPID, SELECTIVE FUJI PHOTO FILM CO., LTD. (JP) 1988-06-14 US disclosed
EP-0025659-B1 PROCESSES FOR THE PRODUCTION OF 1,2,3-TRIHYDROXYPHENYL COMPOUNDS FBC LIMITED (GB) 1983-11-02 EP disclosed
US-4351968-A Production of organic compounds FBC LIMITED (GB) 1982-09-28 US disclosed
EP-0025659-A2 Processes for the production of 1,2,3-trihydroxyphenyl compounds FBC LIMITED (GB) 1981-03-25 EP disclosed
US-4069340-A ARYLOXY DIMETHYL IMMONIUM CHLORIDES FROM DIMETHYL FORMAMIDE AND CORRESPONDING ARYL CHLOROFORMATES HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1978-01-17 US disclosed
US-3983178-A Immonium salts and derivatives thereof HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1976-09-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190343842-A1 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS SIK1, SIK3, SIK2 L3MBTL1 4559/4885SMN1; SMN2 4139/4885ALDH1A1 3380/4885
US-20200338087-A9 USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS SIK1, SIK3, SIK2 L3MBTL1 4559/4885SMN1; SMN2 4139/4885ALDH1A1 3380/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.