SCHEMBL10523979

SCHEMBL10523979

Cc1cccc(C)c1OC(N)=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
ATM Q13315 1/20 0.45
PTPN1 P18031 1/20 0.42
TSHR P16473 3/20 0.41
SCN4A P35499 3/20 0.39
LMNA P02545 2/20 0.39
SCN1A P35498 2/20 0.39
SCN5A Q14524 2/20 0.39
SCN9A Q15858 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29728559 0.88 PTPN1 (0.49) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL29728542 0.86 MEN1 (0.43) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL27641372 0.85 TSHR (0.49) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL28709713 0.82 KDM4E (0.54) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL8764787 0.81 L3MBTL1 (0.55) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL28611098 0.80 TDP1 (0.53) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL982574 0.79 L3MBTL1 (0.58) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL2059537 0.79 KDM4E (0.71) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1
SCHEMBL1951034 0.77 KDM4E (0.41) KMT2AMEN1ALDH1A1KDM4ELMNA
SCHEMBL10959076 0.77 L3MBTL1 (0.52) L3MBTL1SMN1; SMN2KMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230192613-A1 Charged Ion Channel Blockers and Methods for Use NOCION THERAPEUTICS INC (US) 2023-06-22 US disclosed
CN-112020493-B Method for producing urethane and method for producing isocyanate 旭化成株式会社 2023-04-21 CN disclosed
US-11603355-B2 Charged ion channel blockers and methods for use Nocion Therapeutics, Inc. (US) 2023-03-14 US disclosed
EP-3938345-A1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE Nocion Therapeutics, Inc. (US) 2022-01-19 EP disclosed
CN-113950471-A Charged ion channel blockers and methods of use thereof 诺西恩医疗公司 2022-01-18 CN disclosed
US-10968179-B2 Charged ion channel blockers and methods for use Nocion Therapeutics, Inc. (US) 2021-04-06 US disclosed
US-20210061763-A1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE NOCION THERAPEUTICS INC (US) 2021-03-04 US disclosed
US-20200290953-A1 Charged Ion Channel Blockers and Methods for Use Nocion Therapeutics, Inc. 2020-09-17 US disclosed
WO-2020185830-A1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE Nocion Therapeutics, Inc. (US) 2020-09-17 WO disclosed
EP-2755949-B1 FUNGICIDAL 4-SUBSTITUTED-3-{PHENYL[(HETEROCYCLYLMETHOXY)IMINO]METHYL}-1,2,4-OXADIZOL-5(4H)-ONE DERIVATIVES BAYER IP GMBH (DE) 2015-10-21 EP disclosed
US-9090600-B2 Fungicidal 4-substituted-3-{phenyl[(heterocyclylmethoxy)imino]methyl}-1,2,4-oxadizol-5(4H)-one derivatives BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-28 US disclosed
US-20140349848-A1 FUNGICIDAL 4-SUBSTITUTED-3--1,2,4-OXADIZOL-5(4H)-ONE DERIVATIVES BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-11-27 US disclosed
EP-0325620-A1 METHOD FOR THE PREPARATION OF AMIDINO-UREA DERIVATIVES REANAL FINOMVEGYSZERGYAR (HU) 1989-08-02 EP disclosed
WO-1988007990-A1 METHOD FOR THE PREPARATION OF AMIDINO-UREA DERIVATIVES REANAL FINOMVEGYSZERGYÁR (HU) 1988-10-20 WO disclosed
US-4226883-A Carbamate derivatives and method for manufacture thereof YAMAMOTO IZURU 1980-10-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200290953-A1 Charged Ion Channel Blockers and Methods for Use TRPV1, TRPV2, TRPV5 L3MBTL1 4844/4885SMN1; SMN2 2763/4885KMT2A 2429/4885
US-20140349848-A1 FUNGICIDAL 4-SUBSTITUTED-3--1,2,4-OXADIZOL-5(4H)-ONE DERIVATIVES CYP4X1, CYP4B1, CYP4Z1 L3MBTL1 499/4885SMN1; SMN2 1570/4885KMT2A 2404/4885
US-11603355-B2 Charged ion channel blockers and methods for use TRPV1, TRPV2, TRPV5 L3MBTL1 4844/4885SMN1; SMN2 2763/4885KMT2A 2429/4885
US-20230192613-A1 Charged Ion Channel Blockers and Methods for Use TRPV1, TRPV2, TRPV5 L3MBTL1 4844/4885SMN1; SMN2 2763/4885KMT2A 2429/4885
US-10968179-B2 Charged ion channel blockers and methods for use TRPV1, TRPV2, TRPV5 L3MBTL1 4844/4885SMN1; SMN2 2763/4885KMT2A 2429/4885
US-20210061763-A1 CHARGED ION CHANNEL BLOCKERS AND METHODS FOR USE TRPV1, TRPV2, TRPV5 L3MBTL1 4844/4885SMN1; SMN2 2763/4885KMT2A 2429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.