SCHEMBL481776

SCHEMBL481776

Cc1cc(C(=O)O)ccc1C1OC(C)(C)C(C)(C)O1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
ESR1 P03372 2/20 0.41
MYC P01106 1/20 0.41
ALOX15 P16050 1/20 0.41
PTPN7 P35236 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
TDP1 Q9NUW8 3/20 0.41
GRM1 Q13255 2/20 0.41
CYP1A2 P05177 1/20 0.41
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 3/20 0.38
GAA P10253 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
RXRA P19793 4/20 0.38
POLB P06746 2/20 0.37
THRB P10828 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL481777 0.78 TSHR (0.37) TSHRESR1MYCALOX15PTPN7
SCHEMBL9946130 0.75 KMO (0.49) TSHRMYCALOX15PTPN7HSD17B10
SCHEMBL488607 0.74 TSHR (0.46) TSHRALOX15MEN1KMT2ATDP1
SCHEMBL10148368 0.73 CREBBP (0.50) TSHRESR1MYCALOX15PTPN7
SCHEMBL11894061 0.72 TDP1 (0.43) TSHRESR1MYCALOX15PTPN7
SCHEMBL28754473 0.71 RXRB (0.39) ESR1MYCHSD17B10MEN1KMT2A
SCHEMBL4946903 0.70 KMO (0.54) TSHRESR1MYCALOX15PTPN7
SCHEMBL4951622 0.69 KMO (0.57) TSHRESR1MYCALOX15PTPN7
SCHEMBL29421064 0.68 CES2 (0.63) TSHRESR1MYCALOX15PTPN7
SCHEMBL310259 0.68 CES2 (0.63) TSHRESR1MYCALOX15PTPN7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078016-B1 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARM LLC (US) 2012-02-01 EP disclosed