SCHEMBL4818708

SCHEMBL4818708

CCOc1cc(-c2cccc(N(c3ccnc(-n4c(C)ccc4C)c3)c3cc(O)c(OCc4ccccc4)cc3OC)n2)c(OC)cc1OCCN(C)C

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.41
NOS3 P29474 3/20 0.41
EGFR P00533 1/20 0.31
NOS2 P35228 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
PTGER1 P34995 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424624 0.81 NOS1 (0.57) NOS1NOS3EGFRNOS2MEN1
Ammonia Solution, Strong SCHEMBL253374 0.80 NOS1 (0.44) NOS1NOS3EGFRNOS2MEN1
SCHEMBL253373 0.80 NOS1 (0.42) NOS1NOS3EGFRNOS2MEN1
SCHEMBL4286592 0.72 PTGER1 (0.41) PTGER1
SCHEMBL7077507 0.70 NOS3 (0.43) NOS1NOS3PTGER1
SCHEMBL4286467 0.65 NOS1 (0.89) NOS1NOS3NOS2
SCHEMBL5778138 0.65 NOS1 (0.47) NOS1NOS3PTGER1
SCHEMBL7073841 0.64 KDM4E (0.37) NOS1NOS3PTGER1
SCHEMBL7073102 0.60 NOS1 (1.00) NOS1NOS3NOS2
SCHEMBL6581790 0.60 MAOB (0.44) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910385-A1 BENZOTHIAZOLES AND THIAZOLOPYRIDINES AS SIRTUIN MODULATORS Sirtris Pharmaceuticals, Inc. (US) 2008-04-16 EP disclosed
WO-2007019346-A1 BENZOTHIAZOLES AND THIAZOLOPYRIDINES AS SIRTUIN MODULATORS SIRTRIS PHARMACEUTICALS, INC. (US) 2007-02-15 WO disclosed