SCHEMBL4823142

SCHEMBL4823142

CCN(CC)C(=O)c1cc(-c2ccccc2)[nH]c1C

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.61
ALDH1A1 P00352 5/20 0.50
HPGD P15428 5/20 0.50
MAPT P10636 2/20 0.50
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
CDC7 O00311 1/20 0.44
TDP1 Q9NUW8 1/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
TAS2R38 P59533 1/20 0.41
GAA P10253 1/20 0.40
KEAP1 Q14145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2215320 0.79 BRD4 (0.75) BRD4ALDH1A1MAPTCDC7TAS2R38
SCHEMBL1156069 0.78 BRD4 (0.63) BRD4ALDH1A1HPGDMAPTTSHR
SCHEMBL7173993 0.76 BRD4 (1.00) BRD4ALDH1A1MAPTCDC7
SCHEMBL1450398 0.76 BRD4 (0.71) BRD4ALDH1A1MAPTCDC7TAS2R38
SCHEMBL14134219 0.72 HDAC7 (0.57) ALDH1A1HPGDMAPTTSHRMAPK1
SCHEMBL15444821 0.72 BRD4 (0.63) BRD4ALDH1A1HPGDMAPTCDC7
SCHEMBL14134248 0.72 HPGD (0.51) ALDH1A1HPGDMAPTTSHRMAPK1
SCHEMBL375495 0.71 BRD4 (0.58) BRD4ALDH1A1MAPTTSHRMAPK1
SCHEMBL3629780 0.71 MEN1 (0.66) ALDH1A1HPGDMAPTTSHRMAPK1
SCHEMBL29822323 0.71 TP53 (0.69) ALDH1A1HPGDMAPTTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101346381-A New anti-malaria derivatives of 4-aminoquinoline NEED PHARMACEUTICALS S R L (IT) 2009-01-14 CN disclosed
EP-1937686-A1 NEW ANTI-MALARIA DERIVATIVES OF 4-AMINOQUINOLINE Need Pharmaceuticals S.r.l. (IT) 2008-07-02 EP disclosed
WO-2007045987-A1 NEW ANTI-MALARIA DERIVATIVES OF 4-AMINOQUINOLINE NEED PHARMACEUTICALS S.R.L. (IT) 2007-04-26 WO disclosed