SCHEMBL4829454

SCHEMBL4829454

Cc1noc([C@H](N)Cc2ccc(-c3ccc(F)c(F)c3)cc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
GRIN1 Q05586 4/20 0.39
GRIN2B Q13224 4/20 0.39
DPP4 P27487 4/20 0.38
ROCK2 O75116 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA5 P30532 1/20 0.34
CHRNA4 P43681 1/20 0.34
DPP8 Q6V1X1 1/20 0.34
WNT3A P56704 1/20 0.34
TPH1 P17752 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ACHE P22303 1/20 0.33
PTPN1 P18031 1/20 0.32
HTR1A P08908 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3996630 0.89 DPP4 (0.38) GRIN1GRIN2BDPP4DPP8
SCHEMBL4827765 0.89 DPP4 (0.38) GRIN1GRIN2BDPP4DPP8
Hydrochloric Acid SCHEMBL4831560 0.88 DPP4 (0.37) GRIN2BDPP4DPP8
Hydrochloric Acid SCHEMBL4831555 0.88 DPP4 (0.37) GRIN2BDPP4DPP8
SCHEMBL4832003 0.87 TPH1 (0.43) GRIN1GRIN2BDPP4ROCK2DPP8
SCHEMBL4829650 0.84 SLC6A2 (0.42) DPP4ROCK2CYP1A2ACHEPTPN1
SCHEMBL4823412 0.83 TP53 (0.48)
SCHEMBL4829762 0.83 CYP19A1 (0.43) ROCK2TPH1CYP2C9CYP2C19ACHE
SCHEMBL4827767 0.82 GRM2 (0.41) CYP17A1
Hydrochloric Acid SCHEMBL4829646 0.81 GRM2 (0.40) CYP17A1TPH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use VTVX HOLDINGS I LLC 2005-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use CYP2F1, CYP3A43, PNPO CYP17A1 188/4885CYP11B1 47/4885CYP11B2 46/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.