SCHEMBL4831403

SCHEMBL4831403

CNC(=O)c1ccccc1NC(=O)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 15/20 0.67
PPARG P37231 10/20 0.67
NPC1 O15118 1/20 0.64
ALDH1A1 P00352 1/20 0.64
GLA P06280 1/20 0.64
RAB9A P51151 1/20 0.64
ATM Q13315 1/20 0.64
L3MBTL1 Q9Y468 1/20 0.64
PPARA Q07869 6/20 0.60
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
PPARD Q03181 1/20 0.58
MAPT P10636 1/20 0.57
RECQL P46063 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7292297 0.86 NR1H4 (0.74) NR1H4PPARGNPC1ALDH1A1GLA
SCHEMBL6105957 0.86 NR1H4 (0.78) NR1H4PPARGNPC1ALDH1A1GLA
SCHEMBL5226864 0.85 NR1H4 (0.77) NR1H4PPARGPPARAPPARD
SCHEMBL7302098 0.85 PDCD1 (0.68) NR1H4PPARGNPC1ALDH1A1GLA
SCHEMBL15176770 0.85 NPC1 (0.68) NR1H4PPARGNPC1ALDH1A1GLA
SCHEMBL6108092 0.84 TSHR (0.72) NR1H4PPARGNPC1ALDH1A1GLA
SCHEMBL5223315 0.82 RAB9A (0.73) NR1H4PPARGNPC1ALDH1A1GLA
SCHEMBL29903436 0.82 NR1H4 (0.74) NR1H4PPARGPPARAPPARD
SCHEMBL5223950 0.82 NR1H4 (0.71) NR1H4PPARGNPC1RAB9APPARA
SCHEMBL5223825 0.81 NR1H4 (0.71) NR1H4PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed
US-7459472-B2 Aryl and heteroaryl compounds, compositions, and methods of use TRANSTECH PHARMA, INC. (US) 2008-12-02 US disclosed
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use VTVX HOLDINGS I LLC 2005-03-17 US disclosed
WO-2005014534-A1 ARYL AND HETEROARYL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE TRANSTECH PHARMA, INC. (US) 2005-02-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050059713-A1 Aryl and heteroaryl compounds, compositions, and methods of use CYP2F1, CYP3A43, PNPO NR1H4 423/4885PPARG 977/4885NPC1 488/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.