SCHEMBL483568

SCHEMBL483568

CC(C)(C)C1C[C@H](c2ccc(Oc3ccccc3C#N)cc2)N(C(=O)O)[C@]1(C)C(N)=O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.48
EZH2 Q15910 8/20 0.44
MAPK14 Q16539 4/20 0.40
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
LPAR1 Q92633 1/20 0.38
LPAR5 Q9H1C0 1/20 0.38
CYP3A4 P08684 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
BTK Q06187 1/20 0.35
DHODH Q02127 1/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL483784 0.86 KCNH2 (0.51) KCNH2ALDH1A1
SCHEMBL2837158 0.79 KCNH2 (0.53) KCNH2EZH2MAPK14POLBGAA
SCHEMBL311657 0.79 KCNH2 (0.46) KCNH2NPC1RAB9ATP53
SCHEMBL483795 0.75 KCNH2 (0.54) KCNH2
SCHEMBL310676 0.75 KCNH2 (0.54) KCNH2
SCHEMBL483566 0.74 KCNH2 (0.49) KCNH2EZH2MAPK14POLBGAA
SCHEMBL2835462 0.71 KCNH2 (0.57) KCNH2EZH2MAPK14POLBGAA
SCHEMBL483073 0.70 KCNH2 (0.61) KCNH2EZH2MAPK14POLBGAA
SCHEMBL12973281 0.69 KCNH2 (0.52) KCNH2EZH2MAPK14POLBGAA
SCHEMBL2831512 0.69 KCNH2 (0.47) KCNH2EZH2MAPK14POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153623-B2 Compounds Convergence Pharmaceuticals Limited (GB) 2012-04-10 US disclosed
EP-1934176-B1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LTD (GB) 2012-02-01 EP disclosed