SCHEMBL483784

SCHEMBL483784

CC(C)(C)C1C[C@H](c2ccc(OCc3ccccc3C#N)cc2)N(C(=O)O)[C@]1(C)C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.51
FFAR1 O14842 1/20 0.44
MMP1 P03956 3/20 0.41
ADAM17 P78536 2/20 0.41
MAOB P27338 2/20 0.41
ALKBH1 Q13686 1/20 0.39
ADAMTS4 O75173 1/20 0.39
MMP13 P45452 1/20 0.39
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
SCN3A Q9NY46 5/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
SCN1A P35498 1/20 0.35
SCN4A P35499 1/20 0.35
SCN7A Q01118 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN8A Q9UQD0 1/20 0.35
SCN10A Q9Y5Y9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL483795 0.86 KCNH2 (0.54) KCNH2MAOBSCN3ASCN1ASCN4A
SCHEMBL310676 0.86 KCNH2 (0.54) KCNH2MAOBSCN3ASCN1ASCN4A
SCHEMBL483568 0.86 KCNH2 (0.48) KCNH2ALDH1A1
SCHEMBL483408 0.85 KCNH2 (0.46) KCNH2ADAM17MAOBMMP13
SCHEMBL311657 0.85 KCNH2 (0.46) KCNH2ADAM17MAOBMMP13
SCHEMBL2833719 0.81 KCNH2 (0.55) KCNH2FFAR1MMP1ADAM17MAOB
SCHEMBL483783 0.76 KCNH2 (0.51) KCNH2FFAR1MMP1ADAM17MAOB
SCHEMBL483581 0.73 KCNH2 (0.55) KCNH2ALDH1A1ALOX15SCN3ASCN1A
SCHEMBL483295 0.73 KCNH2 (0.51) KCNH2MAOBSCN3ASCN1ASCN4A
SCHEMBL483705 0.72 KCNH2 (0.63) KCNH2FFAR1MMP1ADAM17MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153623-B2 Compounds Convergence Pharmaceuticals Limited (GB) 2012-04-10 US disclosed
EP-1934176-B1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LTD (GB) 2012-02-01 EP disclosed