SCHEMBL4842810

SCHEMBL4842810

CCCc1nc(N)nc2ccc(-c3cccc(C(=O)OCC)c3)nc12.CCCc1nc(N)nc2ccc(-c3ccccc3C(=O)OCC)nc12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.42
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
CCR6 P51684 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
TP53 P04637 1/20 0.38
BRAF P15056 1/20 0.38
PDE2A O00408 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ERN1 O75460 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4101378 0.92 NPC1 (0.44) HSP90AA1RAB9ANPC1TP53BRAF
SCHEMBL4102052 0.91 HSP90AA1 (0.50) HSP90AA1RAB9ANPC1CCR6KDM4E
SCHEMBL4095683 0.83 DHFR (0.51) RAB9ANPC1MAPTALOX15
SCHEMBL4101913 0.82 TLR8 (0.47) HSP90AA1ALDH1A1HSD17B10
SCHEMBL4107011 0.82 NPC1 (0.47) RAB9ANPC1CCR6ALDH1A1MAPT
SCHEMBL4110201 0.81 HSP90AA1 (0.46) HSP90AA1RAB9ANPC1SMN1; SMN2
SCHEMBL4112827 0.81 MAP4K4 (0.41) KDM4EALDH1A1MAPTGAAHPGD
SCHEMBL4101142 0.80 MAP4K4 (0.44) PDE2A
SCHEMBL4097644 0.80 KDM4E (0.37) HSP90AA1KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL4107871 0.80 ALDH1A1 (0.42) HSP90AA1RAB9ANPC1CCR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed