SCHEMBL4844841

SCHEMBL4844841

Cc1cc(O)nc2c1c(OC(=O)ON1CCC(C)CC1)nn2C(=O)N1CCC(C(F)(F)F)CC1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HTT P42858 1/20 0.32
RAB9A P51151 1/20 0.32
SPR P35270 7/20 0.32
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4844815 0.91 SPR (0.30) SPR
SCHEMBL2962458 0.89 GAA (0.35) HPGDSMN1; SMN2HTTRAB9ASPR
SCHEMBL1573996 0.85 SPR (0.35) SPR
SCHEMBL16242498 0.84 HPGD (0.35) HPGDSMN1; SMN2HTTRAB9A
SCHEMBL1573805 0.81 HRH3 (0.35) SPR
SCHEMBL1573736 0.77 SPR (0.35) HPGDSPR
SCHEMBL16242496 0.76 SPR (0.32) HPGDSMN1; SMN2HTTRAB9ASPR
SCHEMBL4833062 0.75 PDE10A (0.35) SPR
SCHEMBL16242494 0.74 TRPV1 (0.34) HPGD
SCHEMBL16242373 0.73 HPGD (0.34) HPGDSMN1; SMN2HTTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937648-B1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI SA (FR) 2014-11-26 EP disclosed
EP-1937648-A1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS sanofi-aventis (FR) 2008-07-02 EP disclosed
WO-2007042178-A1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI-AVENTIS (DE) 2007-04-19 WO disclosed