SCHEMBL4844815

SCHEMBL4844815

Cc1cc(O)nc2c1c(OC(=O)ON1CCC(C(F)(F)F)CC1)nn2C(=O)N1CCN(C)CC1

nearest known ligand 0.30

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
SPR P35270 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4844841 0.91 HPGD (0.32) SPR
SCHEMBL1573805 0.89 HRH3 (0.35) SPR
SCHEMBL1573996 0.84 SPR (0.35) SPR
SCHEMBL2962458 0.80 GAA (0.35) SPR
SCHEMBL4833062 0.75 PDE10A (0.35) SPR
SCHEMBL1573736 0.75 SPR (0.35) SPR
SCHEMBL4828449 0.69 SPR (0.34) SPR
SCHEMBL16242496 0.67 SPR (0.32) SPR
SCHEMBL16242494 0.65 TRPV1 (0.34)
SCHEMBL1573785 0.64 SPR (0.37) SPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937648-B1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI SA (FR) 2014-11-26 EP disclosed
EP-1937648-A1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS sanofi-aventis (FR) 2008-07-02 EP disclosed
WO-2007042178-A1 DIACYL INDAZOL DERIVATIVES AS LIPASE AND PHOSPHOLIPASE INHIBITORS SANOFI-AVENTIS (DE) 2007-04-19 WO disclosed