SCHEMBL4844962

SCHEMBL4844962

CCCc1nc(N)nc2ccc(-c3ccc(OC)cc3)nc12.CCCc1nc(N)nc2ccc(-c3cccc(OC)c3)nc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 2/20 0.52
HRH2 P25021 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
DHFR P00374 2/20 0.44
ADORA2A P29274 1/20 0.44
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
TLR8 Q9NR97 2/20 0.42
DYRK1A Q13627 1/20 0.41
TLR7 Q9NYK1 1/20 0.41
HEXA P06865 1/20 0.41
HEXB P07686 1/20 0.41
PIK3CG P48736 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4113326 0.96 MAP4K4 (0.56) MAP4K4DHFRADORA2AALDH1A1HPGD
SCHEMBL4107851 0.91 HRH2 (0.51) HRH2HRH3DHFRADORA2AALDH1A1
SCHEMBL4114967 0.83 NPC1 (0.43) MAP4K4HRH2HRH3DHFRADORA2A
SCHEMBL4114833 0.81 MAOB (0.46) MAP4K4DHFR
SCHEMBL4101904 0.81 CYP1A2 (0.48) MAP4K4DHFRALDH1A1LMNASMN1; SMN2
SCHEMBL4114040 0.81 MAP4K4 (0.54) MAP4K4DHFRADORA2AALDH1A1LMNA
SCHEMBL4106840 0.80 ALDH1A1 (0.43) MAP4K4HRH2HRH3DHFRALDH1A1
SCHEMBL4096146 0.79 MAP4K4 (0.41) MAP4K4HRH2HRH3DHFRMAPT
SCHEMBL4095683 0.79 DHFR (0.51) MAP4K4DHFRMAPTTLR8TLR7
SCHEMBL4107041 0.78 GAA (0.42) ADORA2AALDH1A1LMNAHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009076-A2 SUBSTITUTED PYRIDO(3,2-D)PYRIMIDINES AND PHARMACEUTICAL COMPOSITIONS FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2008-01-24 WO claimed