SCHEMBL4847152

SCHEMBL4847152

C[C@H](N)C(=O)N(c1cccc2ccccc12)[C@@H](C)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMPD2 O60906 1/20 0.44
SIGMAR1 Q99720 4/20 0.41
AKR1B1 P15121 1/20 0.39
PPARG P37231 4/20 0.37
PPARA Q07869 4/20 0.37
SLC1A3 P43003 2/20 0.37
SLC1A2 P43004 2/20 0.37
SLC1A1 P43005 2/20 0.37
ALOX5 P09917 1/20 0.37
METAP2 P50579 1/20 0.37
NR4A1 P22736 1/20 0.37
NR4A2 P43354 1/20 0.37
NR4A3 Q92570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7437007 0.99 SMPD2 (0.43) SMPD2SIGMAR1AKR1B1PPARGPPARA
SCHEMBL5558314 0.85 SIGMAR1 (0.38) SMPD2SIGMAR1AKR1B1PPARGPPARA
SCHEMBL6119288 0.84 SMPD2 (0.47) SMPD2SIGMAR1AKR1B1PPARGPPARA
SCHEMBL6113113 0.84 SMPD2 (0.47) SMPD2SIGMAR1AKR1B1PPARGPPARA
SCHEMBL6113112 0.84 SMPD2 (0.47) SMPD2SIGMAR1AKR1B1PPARGPPARA
SCHEMBL8497763 0.82 SMPD2 (0.40) SMPD2METAP2
SCHEMBL7902575 0.80 ALPI (0.39) SMPD2METAP2
SCHEMBL7052280 0.80 ALPI (0.39) SMPD2METAP2
SCHEMBL4082840 0.79 SMPD2 (0.48) SMPD2SIGMAR1AKR1B1PPARGPPARA
SCHEMBL1697074 0.79 SMPD2 (0.48) SMPD2SIGMAR1AKR1B1PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012112945-A1 USE OF MATRIX METALLOPROTEINASE INHIBITORS TO TREAT TUBERCULOSIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2012-08-23 WO claimed
US-9750789-B2 Use of matrix metalloproteinase inhibitors to treat tuberculosis THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2017-09-05 US disclosed
WO-2012112945-A1 USE OF MATRIX METALLOPROTEINASE INHIBITORS TO TREAT TUBERCULOSIS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2012-08-23 WO disclosed
EP-1986657-A2 METHOD OF TREATING A SUBJECT SUFFERING FROM DEGENERATIVE DISC DISEASE USING A MATRIX METALLOPROTEASE INHIBITOR Discogen, LLC (US) 2008-11-05 EP disclosed
WO-2007098099-A2 METHOD OF TREATING A SUBJECT SUFFERING FROM DEGENERATIVE DISC DISEASE USING A MATRIX METALLOPROTEASE INHIBITOR DISCOGEN, LLC (US) 2007-08-30 WO disclosed