SCHEMBL7902575

SCHEMBL7902575

CC(C(=O)O)N(C(=O)C(N)Cc1ccc(Br)cc1)c1cccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPI P09923 1/20 0.39
PKM P14618 1/20 0.39
PTGS1 P23219 1/20 0.39
XIAP P98170 1/20 0.39
SLC7A5 Q01650 1/20 0.39
SMPD2 O60906 1/20 0.38
ACACB O00763 2/20 0.38
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
AKT3 Q9Y243 1/20 0.36
LTA4H P09960 1/20 0.35
MME P08473 2/20 0.35
ACP3 P15309 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
GRIK1 P39086 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7052280 1.00 ALPI (0.39) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL4847152 0.80 SMPD2 (0.44) SMPD2METAP2
SCHEMBL8497763 0.79 SMPD2 (0.40) SMPD2KMT2AMMEALDH1A1METAP2
Hydrochloric Acid SCHEMBL7437007 0.79 SMPD2 (0.43) SMPD2METAP2
SCHEMBL6119288 0.76 SMPD2 (0.47) SMPD2
SCHEMBL6113112 0.76 SMPD2 (0.47) SMPD2
SCHEMBL6113113 0.76 SMPD2 (0.47) SMPD2
SCHEMBL10883595 0.73 ALPI (0.56) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL9003246 0.73 SMPD2 (0.45) SMPD2MEN1KMT2AALDH1A1
SCHEMBL29066984 0.72 SLC7A5 (0.55) ALPIPKMPTGS1XIAPSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235717-B1 Pharmaceutical compounds GLAXO WELLCOME INC. 2001-05-22 US disclosed
EP-0677059-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-10-18 EP disclosed
WO-1994015956-A1 ENDOTHELIN CONVERTING ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-07-21 WO disclosed