SCHEMBL4847371

SCHEMBL4847371

CN(C)CCOc1ccccc1C(=O)C=Cc1cccc(CN(C)C)c1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.52
BCHE P06276 6/20 0.50
ACHE P22303 4/20 0.50
HRH1 P35367 1/20 0.47
MAOA P21397 1/20 0.44
ABCG2 Q9UNQ0 1/20 0.44
HSP90AA1 P07900 1/20 0.43
CCR6 P51684 1/20 0.43
HDAC4 P56524 1/20 0.43
MEF2D Q14814 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4857311 0.88 BCHE (0.47) BCHEACHEHRH1
SCHEMBL4853880 0.88 BCHE (0.47) BCHEACHEHRH1
SCHEMBL4853318 0.87 MAOB (0.62) MAOBBCHEACHEMAOA
SCHEMBL5915415 0.86 ABCG2 (0.61) MAOBACHEMAOAABCG2
SCHEMBL25202533 0.86 BCHE (0.65) MAOBBCHEACHEHRH1MAOA
SCHEMBL4856397 0.85 SLC6A9 (0.47) MAOBBCHEACHEHRH1
SCHEMBL4854959 0.85 SLC6A9 (0.47) MAOBBCHEACHEHRH1
SCHEMBL4846158 0.84 BCHE (0.41) MAOBBCHEACHEHRH1HDAC4
SCHEMBL4854696 0.84 BCHE (0.41) MAOBBCHEACHEHRH1HDAC4
SCHEMBL4848357 0.80 MAOB (0.60) MAOBBCHEACHEMAOAABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed