SCHEMBL4847751

SCHEMBL4847751

COc1ccc(/C=C/C(=O)c2cc(-c3cc(C)cc(C)c3)ccc2OCCN(C)C)cc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TUBB1 Q9H4B7 5/20 0.51
TNFRSF1A P19438 2/20 0.51
BCHE P06276 3/20 0.46
ACHE P22303 2/20 0.46
MCL1 Q07820 1/20 0.44
TUBB4A P04350 2/20 0.43
TUBB P07437 2/20 0.43
TUBA3C P0DPH7 2/20 0.43
TUBA1B P68363 2/20 0.43
TUBA4A P68366 2/20 0.43
TUBB4B P68371 2/20 0.43
TUBB3 Q13509 2/20 0.43
TUBB2A Q13885 2/20 0.43
TUBB8 Q3ZCM7 2/20 0.43
TUBA3E Q6PEY2 2/20 0.43
TUBA1A Q71U36 2/20 0.43
TUBA1C Q9BQE3 2/20 0.43
TUBB6 Q9BUF5 2/20 0.43
TUBB2B Q9BVA1 2/20 0.43
SYK P43405 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847787 1.00 TUBB1 (0.51) TUBB1TNFRSF1ABCHEACHEMCL1
SCHEMBL4847316 0.91 MCL1 (0.48) TUBB1TNFRSF1ABCHEACHEMCL1
SCHEMBL4851370 0.91 MCL1 (0.48) TUBB1TNFRSF1ABCHEACHEMCL1
SCHEMBL4847824 0.89 TUBB1 (0.55) TUBB1TNFRSF1ABCHEACHEMCL1
SCHEMBL4853445 0.89 TUBB1 (0.55) TUBB1TNFRSF1ABCHEACHEMCL1
SCHEMBL4847429 0.89 BCHE (0.46) TNFRSF1ABCHEACHESYKMEN1
SCHEMBL4849953 0.89 BCHE (0.46) TNFRSF1ABCHEACHESYKMEN1
SCHEMBL6141442 0.89 MAOA (0.46) TUBB1BCHEACHETUBB4ATUBB
SCHEMBL4856235 0.89 MAOA (0.46) TUBB1BCHEACHETUBB4ATUBB
SCHEMBL4854085 0.88 ABCG2 (0.51) TNFRSF1ABCHEACHEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed