SCHEMBL4848103

SCHEMBL4848103

CN(C)CCOc1ccc(-c2ccccc2Cl)cc1C(=O)/C=C/c1ccccc1CN(C)C

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 8/20 0.47
PTGER1 P34995 2/20 0.41
PTGER4 P35408 2/20 0.41
PTGER3 P43115 2/20 0.41
PTGER2 P43116 2/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
HRH1 P35367 1/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852269 1.00 SLC6A9 (0.47) SLC6A9PTGER1PTGER4PTGER3PTGER2
SCHEMBL4852999 0.91 PTGER1 (0.41) SLC6A9PTGER1PTGER4PTGER3PTGER2
SCHEMBL4854201 0.91 PTGER1 (0.41) SLC6A9PTGER1PTGER4PTGER3PTGER2
SCHEMBL4852630 0.91 ALDH1A1 (0.41) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH1
SCHEMBL4851088 0.91 ALDH1A1 (0.41) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH1
SCHEMBL4847435 0.90 SLC6A9 (0.46) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH1
SCHEMBL4853595 0.90 AR (0.41) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH1
SCHEMBL4857272 0.90 AR (0.41) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH3
SCHEMBL4854710 0.90 AR (0.41) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH1
SCHEMBL4848069 0.90 AR (0.41) SLC6A9KDM4EALDH1A1SMN1; SMN2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed