SCHEMBL4851340

SCHEMBL4851340

Cc1ccc(C)c(Cc2nc(C=O)nn2-c2ccc(S(N)(=O)=O)cc2F)c1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.38
PTGES O14684 1/20 0.36
CA2 P00918 12/20 0.34
CA1 P00915 9/20 0.34
CA7 P43166 3/20 0.34
CA9 Q16790 5/20 0.34
CA12 O43570 3/20 0.34
PTGS1 P23219 2/20 0.34
HTT P42858 1/20 0.32
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CA5B Q9Y2D0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4796038 0.91 PTGS2 (0.37) PTGS2PTGESCA2CA1CA7
SCHEMBL3111940 0.88 PTGS2 (0.40) PTGS2PTGESCA2CA1CA7
SCHEMBL4846638 0.85 PTGS2 (0.38) PTGS2PTGESCA2CA1CA7
SCHEMBL14163083 0.85 LMNA (0.39)
SCHEMBL14163058 0.85 PTGS2 (0.38) PTGS2PTGESCA2CA1CA7
SCHEMBL14163144 0.85 PTGS2 (0.38) PTGS2PTGESCA2CA1CA7
SCHEMBL3113686 0.85 PTGS2 (0.38) PTGS2PTGESCA2CA1CA7
SCHEMBL14163189 0.83
SCHEMBL14163190 0.83 PTGS2 (0.36) PTGS2PTGESCA2CA1CA7
SCHEMBL4738254 0.83 PTGS2 (0.36) PTGS2PTGESCA2CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008075152-A1 1- [4- (SULFONYL) -PHENYL] -5- (BENZYL) -IH-I, 2, 4-TRIAZOL DERIVATIVES AS INHIBITORS OF CARBONIC ANHYDRASE FOR TREATING GLAUCOMA OR OCULAR HYPERTENSION PFIZER PRODUCTS INC. (US) 2008-06-26 WO disclosed
WO-2008075152-A1 1- [4- (SULFONYL) -PHENYL] -5- (BENZYL) -IH-I, 2, 4-TRIAZOL DERIVATIVES AS INHIBITORS OF CARBONIC ANHYDRASE FOR TREATING GLAUCOMA OR OCULAR HYPERTENSION PFIZER PRODUCTS INC. (US) 2008-06-26 WO disclosed