Thiamiprine

Thiamiprine

SCHEMBL4852

Cn1cnc([N+](=O)[O-])c1Sc1nc(N)nc2[nH]cnc12

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.56
MAPT P10636 8/20 0.55
HBB P68871 2/20 0.55
LMNA P02545 2/20 0.55
GMNN O75496 1/20 0.55
TP53 P04637 1/20 0.55
PGR P06401 1/20 0.55
CYP3A4 P08684 1/20 0.55
SLC6A4 P31645 1/20 0.55
BLM P54132 1/20 0.55
PMP22 Q01453 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HTT P42858 2/20 0.53
ALDH1A1 P00352 6/20 0.48
RAB9A P51151 1/20 0.47
HPGD P15428 2/20 0.47
GFER P55789 3/20 0.46
CYP2C19 P33261 2/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiamiprine SCHEMBL29350246 1.00 CYP1A2 (0.56) CYP1A2MAPTHBBLMNAGMNN
Azathioprine SCHEMBL3261116 0.85 MAPT (0.68) CYP1A2MAPTHBBLMNAGMNN
Thiamiprine SCHEMBL4851 0.82 MAPT (0.71) CYP1A2MAPTHBBLMNAGMNN
Thiamiprine SCHEMBL670566 0.81 CYP1A2 (0.45) CYP1A2MAPTHBBLMNAGMNN
SCHEMBL13742750 0.79 HBB (0.60) CYP1A2MAPTHBBLMNAGMNN
Thiamiprine SCHEMBL28095327 0.76 MAPT (0.53) CYP1A2MAPTHBBLMNAGMNN
Thiamiprine SCHEMBL15284276 0.74 MAPT (0.59) CYP1A2MAPTHBBLMNAGMNN
Thiamiprine SCHEMBL27866409 0.72 MAPT (0.47) CYP1A2MAPTHBBLMNAGMNN
Azathioprine SCHEMBL4436347 0.71 MAPT (1.00) MAPTHBBLMNAGMNNTP53
Azathioprine SCHEMBL4278 0.71 MAPT (1.00) MAPTHBBLMNAGMNNTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 31061 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4698185-A1 METHODS AND SYSTEMS FOR IMPROVING ANTI-CANCER THERAPIES Osasuna Therapeutics SA (CH) 2026-02-25 EP claimed
EP-4694909-A1 METHODS OF MODULATING THE EPITHELIAL-MESENCHYMAL TRANSITION RS Oncology, LLC (US) 2026-02-18 EP claimed
EP-4688871-A1 SITE-SPEICFIC ORTHOGONAL BIOCONJUGATE MODALITY AND APPLICATION THEREOF Genequantum Healthcare (Suzhou) Co., Ltd. (CN) 2026-02-11 EP claimed
EP-4687999-A1 TROP2 CONJUGATED BIOLOGICAL MOLECULES, PHARMACEUTICAL COMPOSITIONS AND METHODS OBI Pharma, Inc. (TW) 2026-02-11 EP claimed
WO-2000061549-A2 PHARMACEUTICAL COMPOUNDS NICOX S.A. (FR) 2000-10-19 WO claimed
WO-2000061537-A2 PHARMACEUTICAL COMPOUNDS NICOX S.A. (FR) 2000-10-19 WO claimed
WO-2000061541-A2 PHARMACEUTICAL COMPOUNDS NICOX S.A. (FR) 2000-10-19 WO claimed
WO-2000054795-A1 COMBINED THERAPY WITH A CHEMOTHERAPEUTIC AGENT AND AN ONCOLYTIC VIRUS FOR KILLING TUMOR CELLS IN A SUBJECT THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2000-09-21 WO claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-1999058126-B1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES ENDOWMENT RES INHUMAN BIOLOGY (US) 2000-02-17 WO claimed
WO-1999058126-A1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1999-11-18 WO claimed
EP-0641193-A4 CHEMOTHERAPEUTIC DRUG COMBINATIONS. MARTIN DANIEL S (US) 1995-09-06 EP claimed
EP-0641193-A1 CHEMOTHERAPEUTIC DRUG COMBINATIONS PRO-NEURON, INC. (US) 1995-03-08 EP claimed
WO-1993023014-A1 CHEMOTHERAPEUTIC DRUG COMBINATIONS MARTIN DANIEL S (US) 1993-11-25 WO claimed