SCHEMBL4852241

SCHEMBL4852241

CCOc1ccccc1C(=O)C=Cc1cc(-c2ccccc2C)ccc1OCCN(C)C

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.45
AR P10275 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
ATM Q13315 1/20 0.41
HRH1 P35367 1/20 0.40
ESR1 P03372 1/20 0.40
HTR7 P34969 1/20 0.40
PTPN11 Q06124 1/20 0.39
CAPN1 P07384 1/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
MAOB P27338 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
XDH P47989 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852236 0.93 AR (0.48) SLC6A9ARSMN1; SMN2ALDH1A1KDM4E
SCHEMBL4853461 0.93 AR (0.48) SLC6A9ARSMN1; SMN2ALDH1A1KDM4E
SCHEMBL4853942 0.88 AR (0.45) SLC6A9ARSMN1; SMN2ALDH1A1KDM4E
SCHEMBL4847450 0.87 SLC6A9 (0.43) SLC6A9SMN1; SMN2ALDH1A1KDM4EHRH1
SCHEMBL4854695 0.84 SLC6A9 (0.43) SLC6A9SMN1; SMN2ALDH1A1KDM4EHRH1
SCHEMBL4850165 0.83 TNFRSF1A (0.48) SLC6A9ALDH1A1HTR7BCHEACHE
SCHEMBL4849810 0.83 ABCB1 (0.43) SLC6A9ARSMN1; SMN2ALDH1A1KDM4E
SCHEMBL4848410 0.83 SLC6A9 (0.40) SLC6A9SMN1; SMN2ALDH1A1KDM4EHRH1
SCHEMBL4880575 0.83 SLC6A9 (0.40) SLC6A9SMN1; SMN2ALDH1A1KDM4EHRH1
SCHEMBL4853580 0.83 SLC6A9 (0.40) SLC6A9SMN1; SMN2ALDH1A1KDM4EHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed