SCHEMBL4852365

SCHEMBL4852365

Cc1ccccc1-c1ccc(C(=O)C=Cc2ccccc2CN(C)C)c(OCCN(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 2/20 0.41
SLC6A9 P48067 2/20 0.41
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
ESR1 P03372 1/20 0.38
KDR P35968 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.37
HTR7 P34969 1/20 0.37
AR P10275 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
NMT2 O60551 1/20 0.36
NMT1 P30419 1/20 0.36
DRD2 P14416 1/20 0.35
DRD1 P21728 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4854182 1.00 HRH1 (0.41) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4847435 0.93 SLC6A9 (0.46) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4853568 0.93 SLC6A9 (0.46) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4852369 0.89 HRH1 (0.41) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4847450 0.88 SLC6A9 (0.43) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4856457 0.87 SLC6A9 (0.43) HRH1SLC6A9ALDH1A1KDM4EBCHE
SCHEMBL4854469 0.87 SLC6A9 (0.43) HRH1SLC6A9ALDH1A1KDM4EBCHE
SCHEMBL4854689 0.86 SLC6A9 (0.46) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4855044 0.86 SLC6A9 (0.46) HRH1SLC6A9ALDH1A1KDM4ESMN1; SMN2
SCHEMBL4850218 0.86 SLC6A9 (0.44) SLC6A9ALDH1A1KDM4ESMN1; SMN2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed