SCHEMBL4854769

SCHEMBL4854769

Cc1cc(C)cc(-c2ccc(OCCN(C)C)c(C(=O)/C=C/c3cccc(NCCN(C)C)c3)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SYK P43405 3/20 0.45
BCHE P06276 8/20 0.44
ACHE P22303 7/20 0.44
HCRTR2 O43614 1/20 0.38
MAOB P27338 1/20 0.38
SLC6A9 P48067 1/20 0.38
KDR P35968 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CYSLTR2 Q9NS75 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4852884 1.00 SYK (0.45) SYKBCHEACHEHCRTR2MAOB
SCHEMBL4847745 0.90 SYK (0.47) SYKBCHEACHEMAOB
SCHEMBL4853606 0.90 SYK (0.47) SYKBCHEACHEMAOB
SCHEMBL4853337 0.87 SYK (0.44) SYKBCHEACHEMAOBSLC6A9
SCHEMBL4853507 0.87 MAOA (0.44) SYKBCHEACHEMAOBSLC6A9
SCHEMBL4857314 0.87 MAOA (0.44) SYKBCHEACHEMAOBSLC6A9
SCHEMBL4854231 0.86 BCHE (0.54) SYKBCHEACHESLC6A9
SCHEMBL4853732 0.86 BCHE (0.54) SYKBCHEACHESLC6A9
SCHEMBL4857214 0.85 SYK (0.44) SYKBCHEACHEMAOBSLC6A9
SCHEMBL4856632 0.85 SYK (0.44) SYKBCHEACHEMAOBSLC6A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed