SCHEMBL485722

SCHEMBL485722

O=C(Oc1nccc2cc(N3CCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCCC4(CCNC4)CC3)ccc12)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.38
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
USP28 Q96RU2 2/20 0.34
PIM1 P11309 1/20 0.34
MCHR1 Q99705 1/20 0.34
USP25 Q9UHP3 1/20 0.34
CYP11B1 P15538 1/20 0.33
ALK Q9UM73 1/20 0.33
KHK P50053 1/20 0.33
ALDH1A1 P00352 3/20 0.32
CYP3A4 P08684 3/20 0.32
CYP2D6 P10635 2/20 0.32
TSHR P16473 2/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
IDH1 O75874 1/20 0.32
NPY2R P49146 1/20 0.32
CCR4 P51679 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL484754 0.95 SOS1 (0.39) SOS1SLC6A2SLC6A4SLC6A3USP28
Trifluoroacetic Acid SCHEMBL484753 0.70 MMP2 (0.44) SOS1SLC6A2SLC6A4SLC6A3PIM1
SCHEMBL484729 0.67 SLC6A2 (0.45) SOS1SLC6A2SLC6A4SLC6A3PIM1
SCHEMBL13131256 0.66 SLC6A2 (0.44) SOS1SLC6A2SLC6A4SLC6A3PIM1
SCHEMBL13131249 0.65 CYP11B1 (0.51) SLC6A2SLC6A4SLC6A3PIM1CYP11B1
Hydrochloric Acid SCHEMBL2816087 0.65 SLC6A2 (0.44) SOS1SLC6A2SLC6A4SLC6A3PIM1
SCHEMBL485117 0.64 CYP2D6 (0.51) SOS1SLC6A2SLC6A4SLC6A3MCHR1
SCHEMBL6859491 0.63 CNR2 (0.52) CYP3A4TSHRCYP2C19
Trifluoroacetic Acid SCHEMBL2816008 0.63 HRH4 (0.49) PIM1MCHR1CYP11B1ALDH1A1CYP3A4
Trifluoroacetic Acid SCHEMBL8511708 0.62 HDAC1 (0.39) SLC6A2SLC6A4SLC6A3ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411381-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-02-01 EP disclosed
WO-2010108651-A1 SUBSTITUTED SPIRO-AMIDE COMPOUNDS Grünenthal GmbH (DE) 2010-09-30 WO disclosed